SCHEMBL9749414

SCHEMBL9749414

NNC(=S)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
KIF11 P52732 1/20 0.46
ALDH1A1 P00352 3/20 0.44
MAPT P10636 1/20 0.44
PTGS1 P23219 3/20 0.43
SRD5A2 P31213 1/20 0.42
IDO1 P14902 1/20 0.42
LMNA P02545 1/20 0.42
PTPN1 P18031 2/20 0.42
GSK3B P49841 2/20 0.41
NPC1 O15118 1/20 0.41
CRHBP P24387 1/20 0.41
RAB9A P51151 1/20 0.41
CRHR2 Q13324 1/20 0.41
MMP1 P03956 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
PAX8 Q06710 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4984479 0.79 HDAC1 (0.48) ALDH1A1MAPTSRD5A2LMNANPC1
SCHEMBL182755 0.77 CES2 (0.61) CES2CES1ALDH1A1MAPTPTGS1
SCHEMBL1753793 0.76 IDO1 (0.52) CES2CES1IDO1RAB9A
SCHEMBL261282 0.76 CES2 (0.54) CES2CES1KIF11ALDH1A1PTGS1
SCHEMBL4399783 0.75 CES2 (0.48) CES2CES1ALDH1A1PTGS1SRD5A2
SCHEMBL10919988 0.75 CES2 (0.58) CES2CES1KIF11ALDH1A1SRD5A2
Hydrochloric Acid SCHEMBL2108579 0.74 IDO1 (0.50) CES2CES1IDO1RAB9A
SCHEMBL20997879 0.73 CES2 (0.47) CES2CES1ALDH1A1PTGS1SRD5A2
Hydrochloric Acid SCHEMBL4394743 0.73 CES2 (0.47) CES2CES1ALDH1A1PTGS1SRD5A2
SCHEMBL28477468 0.73 RAB9A (0.57) KIF11ALDH1A1MAPTLMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0217519-B1 5-MEMBERED HETEROCYCLIC RING ANGIOTENSIN CONVERTING ENZYME INHIBITORS FISONS plc (GB) 1992-02-05 EP disclosed
US-4927822-A HYPOTENSIVE FISONS PLC (GB) 1990-05-22 US disclosed
EP-0217519-A1 5-membered heterocyclic ring angiotensin converting enzyme inhibitors FISONS plc (GB) 1987-04-08 EP disclosed