SCHEMBL9749587

SCHEMBL9749587

NNC(=S)c1ccc2ccccc2c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.52
PLG P00747 1/20 0.52
PLAU P00749 1/20 0.52
KLKB1 P03952 1/20 0.52
KLK1 P06870 1/20 0.52
PRSS1 P07477 1/20 0.52
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
ALDH1A1 P00352 4/20 0.46
ALOX12 P18054 2/20 0.46
MAPT P10636 3/20 0.43
NPC1 O15118 3/20 0.43
KDM4E B2RXH2 3/20 0.43
TDP1 Q9NUW8 2/20 0.43
CYP3A4 P08684 2/20 0.43
HSD17B10 Q99714 2/20 0.43
MEN1 O00255 1/20 0.43
EGFR P00533 1/20 0.43
TP53 P04637 1/20 0.43
PKM P14618 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8161020 0.77 F2 (0.63) F2PLGPLAUKLKB1KLK1
SCHEMBL8157181 0.76 PLAU (0.62) F2PLGPLAUKLKB1KLK1
SCHEMBL1149678 0.76 NPC1 (0.62) CES2CES1ALDH1A1MAPTNPC1
SCHEMBL13377779 0.75 CES2 (0.54) F2PLGPLAUKLKB1KLK1
Hydrochloric Acid SCHEMBL20299655 0.74 NPC1 (0.60) CES2CES1ALDH1A1MAPTNPC1
Hydrochloric Acid SCHEMBL22558263 0.74 HTT (0.54) ALDH1A1MAPTNPC1KDM4ECYP3A4
SCHEMBL1479594 0.74 CES2 (0.58) F2PLGPLAUKLKB1KLK1
SCHEMBL6261300 0.73 ALDH1A1 (0.60) ALDH1A1MAPTKDM4ETDP1CYP3A4
SCHEMBL442250 0.73 POLB (0.50) ALDH1A1ALOX12MAPTNPC1HSD17B10
SCHEMBL16527108 0.72 CES2 (0.56) F2PLGPLAUKLKB1KLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0217519-B1 5-MEMBERED HETEROCYCLIC RING ANGIOTENSIN CONVERTING ENZYME INHIBITORS FISONS plc (GB) 1992-02-05 EP disclosed
US-4927822-A HYPOTENSIVE FISONS PLC (GB) 1990-05-22 US disclosed
EP-0217519-A1 5-membered heterocyclic ring angiotensin converting enzyme inhibitors FISONS plc (GB) 1987-04-08 EP disclosed