SCHEMBL9750264

SCHEMBL9750264

c1ccc2c(c1)N=NNO2

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.33
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
ALOX5 P09917 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3177319 0.98 KDM4E (0.32) TRPA1CYP1A2CYP2D6
SCHEMBL452614 0.76
SCHEMBL11767356 0.69 TRPA1 (0.52) TRPA1CYP1A2CYP2D6ALOX5
SCHEMBL34463644 0.68
SCHEMBL6808163 0.67
SCHEMBL1938763 0.64 TRPA1 (0.42) TRPA1CYP1A2CYP2D6ALOX5
SCHEMBL207166 0.62 TRPA1 (0.32) TRPA1CYP1A2CYP2D6
SCHEMBL9844067 0.59 LMNA (0.41) TRPA1CYP1A2CYP2D6
SCHEMBL5034772 0.59 TRPA1 (0.42) TRPA1ALOX5
SCHEMBL2094585 0.59 TRPA1 (0.42) TRPA1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0219852-B1 CHARTREUSIN DERIVATIVES, SALTS THEREOF, ANTITUMOROUS COMPOSITIONS CONTAINING THE SAME, AND PROCESSES FOR PRODUCING THE SAME ISHIHARA SANGYO KAISHA, LTD. (JP) 1992-02-05 EP disclosed
US-5064945-A Antitumor Agents ISHIHARA SANGYO KAISHA, LTD. (JP) 1991-11-12 US disclosed
US-4927919-A ANTITUMOR AGENTS ISHIHARA SANGYO KAISHA, LTD. (JP) 1990-05-22 US disclosed
EP-0219852-A2 Chartreusin derivatives, salts thereof, antitumorous compositions containing the same, and processes for producing the same ISHIHARA SANGYO KAISHA, LTD. (JP) 1987-04-29 EP disclosed