SCHEMBL9750285

SCHEMBL9750285

C=C1N(CC)c2ccc(OCc3ccccc3)cc2C1(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.43
ALOX5 P09917 1/20 0.42
MAOB P27338 6/20 0.40
MEN1 O00255 2/20 0.40
NPC1 O15118 2/20 0.40
KMT2A Q03164 2/20 0.40
TP53 P04637 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PDK2 Q15119 1/20 0.40
FSHR P23945 1/20 0.40
RAB9A P51151 1/20 0.40
MAOA P21397 2/20 0.39
CYP3A4 P08684 1/20 0.39
SIRT2 Q8IXJ6 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
SIRT5 Q9NXA8 1/20 0.39
BCHE P06276 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9750432 0.85 HRH3 (0.48) HRH3ALOX5MAOBMEN1NPC1
SCHEMBL4615673 0.80 ALDH1A1 (0.45) MEN1KMT2AKDM4EALDH1A1SMN1; SMN2
SCHEMBL11019035 0.77 HRH3 (0.48) HRH3ALOX5MAOBMEN1NPC1
SCHEMBL9893372 0.76 KCNA5 (0.50) ALOX5MAOBTP53MAOASIRT2
SCHEMBL28250868 0.74 POLB (0.48) HRH3ALOX5MAOBMEN1NPC1
SCHEMBL9750274 0.73 MAOB (0.43) HRH3MAOBNPC1SMN1; SMN2RAB9A
SCHEMBL6091601 0.73 KMT2A (0.46) MEN1NPC1KMT2ATP53KDM4E
SCHEMBL9750098 0.72 MAOB (0.46) MAOBMEN1KMT2AMAOA
SCHEMBL9893431 0.72 KCNA5 (0.58)
SCHEMBL9893318 0.72 KCNA5 (0.45) HRH3MAOBTP53MAOASIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120858-A Condensation of 2-methyleneindoline and formic acid in acetic anhydride MILES INC. (US) 1992-06-09 US disclosed
EP-0058863-B1 PROCESS FOR THE PREPARATION OF TRIMETHINE DYESTUFFS BAYER AG (DE) 1985-01-23 EP disclosed
US-4419511-A Process for the preparation of trimethine dyestuffs BAYER AKTIENGESELLSCHAFT (US) 1983-12-06 US disclosed
EP-0058863-A1 Process for the preparation of trimethine dyestuffs BAYER AG (DE) 1982-09-01 EP disclosed