SCHEMBL9750401

SCHEMBL9750401

O=C(O)c1cn(-c2ccc(F)cc2)c2c(F)c(N3CCNCC3CO)c(F)cc2c1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.53
ALDH1A1 P00352 7/20 0.53
HPGD P15428 6/20 0.53
HSD17B10 Q99714 6/20 0.53
LMNA P02545 5/20 0.53
POLB P06746 1/20 0.46
HSP90AA1 P07900 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
PIM1 P11309 3/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
TOP2A P11388 5/20 0.44
TOP2B Q02880 4/20 0.44
TOP1 P11387 1/20 0.44
PMP22 Q01453 1/20 0.43
BRD4 O60885 1/20 0.41
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
CYP2J2 P51589 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9750404 0.90 KDM4E (0.42) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL9749297 0.87 KDM4E (0.50) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL10425974 0.87 KDM4E (0.50) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL9749304 0.86 LMNA (0.53) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL9870203 0.84 KDM4E (0.66) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL9749919 0.84 KDM4E (0.61) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL10426035 0.83 KDM4E (0.61) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL9750386 0.83 KDM4E (0.45) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL9749838 0.83 TOP2A (0.53) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL10372535 0.81 KDM4E (0.62) KDM4EALDH1A1HPGDHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0216345-B1 QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1992-02-19 EP disclosed
US-4977265-A WITH BACTERICIDAL ACTIVITY HOFFMANN-LA ROCHE INC. (US) 1990-12-11 US disclosed
US-4946847-A BACTERICIDES HOFFMANN-LA ROCHE INC. (US) 1990-08-07 US disclosed
US-4806541-A ANTIBACTERIAL AGENTS HOFFMANN-LA ROCHE INC. (US) 1989-02-21 US disclosed
EP-0216345-A2 Quinoline derivatives F. HOFFMANN-LA ROCHE AG (CH) 1987-04-01 EP disclosed