SCHEMBL9751587

SCHEMBL9751587

c1ccc2c(NC3NCCN3)csc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.45
MAPT P10636 7/20 0.42
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
CHRM2 P08172 2/20 0.37
CHRM4 P08173 2/20 0.37
CHRM5 P08912 2/20 0.37
CHRM1 P11229 2/20 0.37
CHRM3 P20309 2/20 0.37
CYP2A6 P11509 3/20 0.37
GAA P10253 1/20 0.36
MAPK1 P28482 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6482190 0.72 PKM (0.58) PKMMAPTRAB9ANPC1CHRM2
SCHEMBL23445461 0.71 PKM (0.46) PKMMAPTRAB9ANPC1CHRM2
SCHEMBL2354792 0.69 PKM (0.59) PKMMAPTRAB9ANPC1CHRM2
Hydrochloric Acid SCHEMBL5357792 0.67 PKM (0.58) PKMMAPTRAB9ANPC1CHRM2
SCHEMBL17887902 0.66 PTGIR (0.54) RAB9ANPC1CHRM2CHRM1SLC6A4
SCHEMBL17740783 0.66 MAPT (0.60) PKMMAPTRAB9ANPC1CYP2A6
SCHEMBL7993430 0.65 SLC6A4 (0.40) MAPTCHRM2CHRM4CHRM5CHRM1
SCHEMBL5805784 0.65 PKM (0.50) PKMMAPTRAB9ANPC1CYP2A6
SCHEMBL277681 0.65 PKM (0.54) PKMMAPTRAB9ANPC1CYP2A6
SCHEMBL8159575 0.64 DDB1 (0.39) PKMMAPTMAPK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422119-A4 BENZOTHIOPHENE DERIVATIVES USEFUL FOR MODIFYING FEEDING BEHAVIOR AND OBSESSIVE-COMPULSIVE BEHAVIOR 1991-11-13 EP disclosed
EP-0422119-A1 BENZOTHIOPHENE DERIVATIVES USEFUL FOR MODIFYING FEEDING BEHAVIOR AND OBSESSIVE-COMPULSIVE BEHAVIOR NEUREX CORPORATION (US) 1991-04-17 EP disclosed
US-4971974-A ANOREXIGENIC AGENTS, BENZO B!THIENO 2,3-C!PYRIDINE COMPOUNDS NEUREX CORPORATION (US) 1990-11-20 US disclosed
WO-1989012447-A1 BENZOTHIOPHENE DERIVATIVES USEFUL FOR MODIFYING FEEDING BEHAVIOR AND OBSESSIVE-COMPULSIVE BEHAVIOR NEUREX CORPORATION (US) 1989-12-28 WO disclosed