SCHEMBL9751959

SCHEMBL9751959

N#CC(C=O)C(=O)Nc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.49
CYP1A2 P05177 1/20 0.48
CYP2C19 P33261 1/20 0.48
GAA P10253 3/20 0.45
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 5/20 0.45
MAPT P10636 5/20 0.45
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
ATM Q13315 2/20 0.45
LMNA P02545 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 1/20 0.45
TP53 P04637 1/20 0.44
EPHX1 P07099 1/20 0.44
TSHR P16473 1/20 0.44
EPHX2 P34913 1/20 0.44
CDK9 P50750 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11344840 0.77 POLB (0.53) POLBCYP1A2CYP2C19GAAKDM4E
SCHEMBL9223095 0.75 ALDH1A1 (0.56) POLBCYP1A2CYP2C19GAAKDM4E
SCHEMBL2782602 0.75 POLB (0.52) POLBCYP1A2CYP2C19GAAKDM4E
SCHEMBL28762296 0.74 POLB (0.65) POLBCYP1A2CYP2C19GAAKDM4E
SCHEMBL1224747 0.73 TDP1 (0.44) POLBCYP2C19GAAALDH1A1MAPT
SCHEMBL22357366 0.73 POLB (0.53) POLBGAAALDH1A1MAPTMEN1
SCHEMBL11382873 0.72 CYP1A2 (0.59) POLBCYP1A2CYP2C19GAAKDM4E
SCHEMBL9819108 0.71 POLB (0.47) POLBCYP1A2CYP2C19GAAKDM4E
SCHEMBL9819309 0.71 GAA (0.58) POLBCYP1A2CYP2C19GAAKDM4E
SCHEMBL8410641 0.70 MEN1 (0.54) POLBCYP1A2CYP2C19GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0423269-A1 HETEROARYL-3-OXO-PROPANENITRILE DERIVATIVES USEFUL IN THE TREATMENT OF RHEUMATOID ARTHRITIS AND OTHER AUTOIMMUNE DISEASES. ERBA CARLO SPA (IT) 1991-04-24 EP claimed