SCHEMBL9753950

SCHEMBL9753950

Cc1c(C(=O)O)nc2c(CCl)cccn12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
GAA P10253 2/20 0.39
ATP4A P20648 4/20 0.37
ATP4B P51164 4/20 0.37
PTGS1 P23219 2/20 0.36
PTGS2 P35354 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HTT P42858 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
NOTUM Q6P988 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CASP1 P29466 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8607290 0.86 ALDH1A1 (0.40) ALDH1A1GAAATP4AATP4BPTGS1
SCHEMBL8608835 0.84 SMN1; SMN2 (0.48) ALDH1A1GAAPTGS1PTGS2CYP1A2
SCHEMBL9923895 0.80 ALDH1A1 (0.51) ALDH1A1GAAPTGS1PTGS2CYP1A2
SCHEMBL6351785 0.79 CYP3A4 (0.49) ATP4AATP4BCYP1A2CYP3A4CYP2D6
SCHEMBL9753914 0.78 SMN1; SMN2 (0.38) ALDH1A1GAAATP4AATP4BCYP1A2
SCHEMBL7853457 0.72 ATP4A (0.61) ATP4AATP4BCYP1A2CYP3A4CYP2D6
SCHEMBL8608772 0.71 SMN1; SMN2 (0.49) ALDH1A1PTGS1PTGS2CYP1A2CYP3A4
SCHEMBL9081296 0.70 KMT2A (0.46) CYP3A4MAPTHPGDSMN1; SMN2HTT
SCHEMBL8352177 0.69 ALDH1A1 (0.68) ALDH1A1GAAPTGS1PTGS2CYP1A2
SCHEMBL10751414 0.65 CYP1A2 (0.47) ALDH1A1ATP4AATP4BCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0436831-A2 Imidazo[1,2-a]pyridinylalkyl compounds for treatment of neurotoxic injury G.D. Searle & Co. (US) 1991-07-17 EP disclosed
WO-1991008211-A1 IMIDAZO[1,2-a]PYRIDINYLALKYL COMPOUNDS FOR TREATMENT OF NEUROTOXIC INJURY G.D. SEARLE & CO. (US) 1991-06-13 WO disclosed