SCHEMBL9754460

SCHEMBL9754460

COc1cccc(-c2cc3ccccc3c3ccccc23)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
BTK Q06187 1/20 0.43
ALDH1A1 P00352 2/20 0.42
HIF1A Q16665 2/20 0.42
HSD17B10 Q99714 2/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
CASP1 P29466 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
CYP11B1 P15538 1/20 0.40
KDR P35968 1/20 0.40
TGFBR1 P36897 1/20 0.39
NISCH Q9Y2I1 1/20 0.38
HSP90AA1 P07900 2/20 0.38
HSP90AB1 P08238 2/20 0.38
TRPM4 Q8TD43 1/20 0.37
IDH1 O75874 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9534117 0.84 ALDH1A1 (0.45) KDM4EBTKALDH1A1HSD17B10HPGD
SCHEMBL16189453 0.79 KDR (0.40) ALDH1A1HSD17B10HPGDMAPK1CYP11B1
SCHEMBL3155981 0.77 BTK (0.61) KDM4EBTKALDH1A1HPGDKDR
SCHEMBL16189114 0.77 ACACA (0.41) KDM4EALDH1A1HSD17B10HPGDTSHR
SCHEMBL10304963 0.75 PDE2A (0.48) BTKALDH1A1HIF1AHSD17B10TSHR
SCHEMBL16225055 0.74 TGFBR1 (0.51) KDM4EBTKALDH1A1HSD17B10TSHR
SCHEMBL21083344 0.74 TGFBR1 (0.48) KDM4EBTKTSHRKDRTGFBR1
SCHEMBL27479812 0.74 BTK (0.44) BTKALDH1A1HSD17B10MAPK1KDR
SCHEMBL14184254 0.74 CYP11B1 (0.47) KDM4EALDH1A1HIF1AHSD17B10HPGD
SCHEMBL9535531 0.72 RAC1 (0.49) KDM4EBTKALDH1A1HPGDKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991017987-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-11-28 WO disclosed