SCHEMBL9754503

SCHEMBL9754503

Cn1c2ccc(C=O)cc2c2sc3ccccc3c21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 3/20 0.43
MAPT P10636 4/20 0.42
RXFP1 Q9HBX9 2/20 0.42
KIF11 P52732 2/20 0.40
TP53 P04637 2/20 0.40
CYP2A6 P11509 1/20 0.37
KDM4E B2RXH2 4/20 0.37
ALDH1A1 P00352 3/20 0.37
AHR P35869 1/20 0.36
NQO2 P16083 1/20 0.35
LMNA P02545 1/20 0.35
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9754492 0.79 MAPT (0.49) MAPTRXFP1TP53KDM4EALDH1A1
SCHEMBL718797 0.75 PTGER4 (0.64) PTGER4MAPTKDM4EALDH1A1NQO2
SCHEMBL29570020 0.75 PTGER4 (0.64) PTGER4MAPTKDM4EALDH1A1NQO2
SCHEMBL17281048 0.74 TP53 (0.43) MAPTRXFP1TP53KDM4EALDH1A1
SCHEMBL17281061 0.73 MAOB (0.43) MAPTRXFP1TP53KDM4EALDH1A1
SCHEMBL13183677 0.72 ALKBH5 (0.50) MAPTRXFP1KIF11TP53KDM4E
SCHEMBL31711447 0.72 CYP2A6 (0.53) PTGER4MAPTKIF11CYP2A6KDM4E
SCHEMBL12170772 0.72 MAPT (0.49) MAPTRXFP1TP53KDM4EALDH1A1
SCHEMBL2713434 0.72 CYP2A6 (0.53) PTGER4MAPTKIF11CYP2A6KDM4E
SCHEMBL6860177 0.71 GPR3 (0.54) MAPTKIF11CYP2A6KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991014688-A1 HETERO POLYCYCLIC BIOCIDAL COMPOUNDS AND THEIR USE IN MEDECINE THE WELLCOME FOUNDATION LIMITED (GB) 1991-10-03 WO disclosed
EP-0447703-A1 Hetero polycyclic biocidal compounds, their synthesis and intermediates therefor,formulations containing them and their use in medicine THE WELLCOME FOUNDATION LIMITED (GB) 1991-09-25 EP disclosed
US-4999369-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-03-12 US disclosed
US-4910218-A With a hydroxy containing secondary amine group BURROUGHS WELLCOME CO. (US) 1990-03-20 US disclosed