SCHEMBL9754832

SCHEMBL9754832

CCCc1nc2c(Br)cccc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
GRM2 Q14416 3/20 0.40
CHEK1 O14757 1/20 0.39
DDAH1 O94760 1/20 0.39
POLB P06746 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
PDE10A Q9Y233 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28871299 0.90 POLB (0.44) ALDH1A1GRM2POLB
SCHEMBL29968130 0.90 POLB (0.44) ALDH1A1GRM2POLB
SCHEMBL31029252 0.86 DDAH1 (0.53) ALDH1A1GRM2CHEK1DDAH1ADORA3
SCHEMBL28871267 0.86 DDAH1 (0.53) ALDH1A1GRM2CHEK1DDAH1ADORA3
SCHEMBL1917210 0.81 MGAM (0.47) ALDH1A1
SCHEMBL28379367 0.81 POLB (0.44) POLBPDE10A
SCHEMBL10397230 0.80 PDE10A (0.57) CHEK1DDAH1POLBKDM4EPDE10A
SCHEMBL1917492 0.80 PSMB8 (0.49) CHEK1DDAH1POLBKDM4EADORA3
SCHEMBL7964155 0.80 CHEK1 (0.58) CHEK1DDAH1POLBKDM4EPDE10A
SCHEMBL31546228 0.80 POLB (0.46) POLBKDM4EPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed
WO-1991013063-A1 NEW BENZIMIDAZOLE DERIVATIVES, METHOD FOR PREPARING THEM AND THEIR PHARMACEUTICAL USE SCHERING AKTIENGESELLSCHAFT BERLIN UND BERGKAMEN (DE) 1991-09-05 WO disclosed