SCHEMBL9757056

SCHEMBL9757056

CCOC(=O)C1Oc2cc(O)cc(O)c2N1c1ccc(OC)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
HTT P42858 1/20 0.39
BLM P54132 1/20 0.39
GAA P10253 1/20 0.39
SLC5A1 P13866 1/20 0.39
SLC5A2 P31639 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
GLO1 Q04760 1/20 0.39
CYP1A1 P04798 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9757022 0.78 CYSLTR1 (0.47)
SCHEMBL24065978 0.66 SMN1; SMN2 (0.60) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL24065915 0.66 SMN1; SMN2 (0.60) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL17977269 0.65 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL8260150 0.65 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL7434354 0.65 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL7436135 0.65 ALDH1A1 (0.53) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL7430439 0.65 ALDH1A1 (0.53) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL7434157 0.65 ALDH1A1 (0.53) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL28535310 0.64 ALDH1A1 (0.55) ALDH1A1KDM4EHPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019475-A2 QUINOLINYL-BENZOHETEROBICYCLIC DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D¿4? RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1991-12-26 WO disclosed
US-5041453-A Quinolinyl-benzoheterobicyclic derivatives as antagonists of leukotriene D4 RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-08-20 US disclosed