SCHEMBL9757080

SCHEMBL9757080

Cc1c(-c2nnn[nH]2)sc2ccc(OCc3ccc(C=Cc4ccc5ccc(Cl)cc5n4)cc3)cc12

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYSLTR1 Q9Y271 7/20 0.35
CYSLTR2 Q9NS75 5/20 0.35
ATP4A P20648 1/20 0.34
ATP4B P51164 1/20 0.34
ROCK1 Q13464 4/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
THRB P10828 1/20 0.33
MAPK1 P28482 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
ATM Q13315 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9757649 0.90 CYSLTR1 (0.44) CYSLTR1CYSLTR2
SCHEMBL9757075 0.82 ROCK1 (0.32) ROCK1KMT2A
SCHEMBL9757146 0.81 TEC (0.37) CYSLTR1CYSLTR2ATP4AATP4BRAB9A
SCHEMBL9757150 0.81 CYSLTR1 (0.43) CYSLTR1CYSLTR2KDM4ENPC1RAB9A
SCHEMBL9757192 0.77 PDE10A (0.51) CYSLTR1CYSLTR2
SCHEMBL9757647 0.76 MAOB (0.34) CYSLTR1CYSLTR2ROCK1
SCHEMBL9757240 0.75 TEC (0.38) CYSLTR1CYSLTR2KDM4EMEN1NPC1
SCHEMBL9757187 0.75 TEC (0.38) CYSLTR1CYSLTR2KDM4EMEN1NPC1
SCHEMBL9756987 0.72 PDE10A (0.49) CYSLTR1CYSLTR2
SCHEMBL9757078 0.71 CYSLTR1 (0.53) CYSLTR1CYSLTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019475-A2 QUINOLINYL-BENZOHETEROBICYCLIC DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D¿4? RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1991-12-26 WO disclosed