SCHEMBL9757130

SCHEMBL9757130

CCOC(=O)c1nc2cc([N+](=O)[O-])c(O)cc2o1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
LMNA P02545 2/20 0.43
POLB P06746 2/20 0.43
MITF O75030 2/20 0.43
GALR2 O43603 1/20 0.43
HSP90AA1 P07900 1/20 0.43
HPGD P15428 1/20 0.43
XBP1 P17861 1/20 0.43
CCR6 P51684 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
GSTP1 P09211 2/20 0.39
GSTM2 P28161 2/20 0.39
KMT2A Q03164 1/20 0.39
MAPT P10636 4/20 0.39
NPC1 O15118 2/20 0.39
PKM P14618 1/20 0.39
CRHBP P24387 1/20 0.39
RAB9A P51151 1/20 0.39
CRHR2 Q13324 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9757163 0.83 CYP3A4 (0.41) ALDH1A1SMN1; SMN2HPGDNPSR1MAPT
SCHEMBL10737642 0.75 HIF1A (0.54) ALDH1A1SMN1; SMN2HPGDNPSR1KMT2A
SCHEMBL9757218 0.75 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2LMNAPOLBMITF
SCHEMBL9197360 0.75 MIF (0.54) ALDH1A1SMN1; SMN2LMNAHPGDKMT2A
SCHEMBL9488561 0.74 ALDH1A1 (0.59) ALDH1A1SMN1; SMN2LMNAPOLBMITF
SCHEMBL3611112 0.73 AGPAT2 (0.49) ALDH1A1SMN1; SMN2POLBHPGDMAPT
SCHEMBL11161951 0.73 DAGLA (0.51) ALDH1A1SMN1; SMN2POLBKMT2AMAPT
SCHEMBL10650222 0.73 NLRP3 (0.48) ALDH1A1SMN1; SMN2LMNAHPGDKMT2A
SCHEMBL10829127 0.73 KDM4E (0.48) ALDH1A1SMN1; SMN2LMNAHPGDKMT2A
SCHEMBL27892480 0.72 MAPT (0.43) ALDH1A1LMNAKMT2AMAPTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019475-A2 QUINOLINYL-BENZOHETEROBICYCLIC DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D¿4? RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1991-12-26 WO disclosed
US-5041453-A Quinolinyl-benzoheterobicyclic derivatives as antagonists of leukotriene D4 RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-08-20 US disclosed