SCHEMBL9757280

SCHEMBL9757280

CCCOC(=O)c1nc2c(O)c(Cl)ccc2o1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.39
ALDH1A1 P00352 6/20 0.39
ESR1 P03372 2/20 0.39
CHRM1 P11229 1/20 0.39
TSHR P16473 1/20 0.39
SLC6A2 P23975 1/20 0.39
KDR P35968 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
KDM4E B2RXH2 2/20 0.39
AGPAT2 O15120 1/20 0.39
LMNA P02545 2/20 0.37
MAOB P27338 2/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 2/20 0.36
TP53 P04637 1/20 0.36
ALOX5 P09917 1/20 0.34
ADORA3 P0DMS8 1/20 0.33
MAPT P10636 1/20 0.33
STAT1 P42224 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9757047 0.90 ALOX5 (0.42) ALDH1A1AGPAT2MAOBNPC1RAB9A
SCHEMBL9757055 0.76 DPP4 (0.43) ALDH1A1TSHRKDM4ETP53
SCHEMBL9757131 0.76 MAOB (0.42) ALDH1A1ESR1TDP1SMN1; SMN2KDM4E
SCHEMBL28667845 0.71 TP53 (0.61) ALDH1A1TDP1SMN1; SMN2KDM4ELMNA
SCHEMBL19636606 0.71 ALDH1A1 (0.50) POLBALDH1A1ESR1CHRM1TSHR
SCHEMBL9635486 0.71 MAOB (0.58) ALDH1A1ESR1CHRM1TSHRSLC6A2
SCHEMBL11197714 0.67 KMT2A (0.51) POLBALDH1A1ESR1TSHRLMNA
SCHEMBL6233680 0.66 ESR1 (0.47) POLBALDH1A1ESR1CHRM1TSHR
SCHEMBL24986639 0.65 S1PR4 (0.47) ALDH1A1ESR1CHRM1TSHRSLC6A2
SCHEMBL7538753 0.65 GAA (0.34) POLBTDP1KDM4EAGPAT2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019475-A2 QUINOLINYL-BENZOHETEROBICYCLIC DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D¿4? RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1991-12-26 WO disclosed
US-5041453-A Quinolinyl-benzoheterobicyclic derivatives as antagonists of leukotriene D4 RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-08-20 US disclosed