SCHEMBL9762662

SCHEMBL9762662

CCOCCn1ccnc1[C@H]1CCCN(C)C1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.55
HRH1 P35367 7/20 0.41
CHRM1 P11229 4/20 0.41
PDK1 Q15118 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK3 Q15120 1/20 0.39
PDK4 Q16654 1/20 0.39
CYP2D6 P10635 2/20 0.35
HTR2A P28223 1/20 0.32
LSS P48449 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM3 P20309 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9761678 1.00 KCNH2 (0.55) KCNH2HRH1CHRM1PDK1PDK2
SCHEMBL9762594 1.00 KCNH2 (0.55) KCNH2HRH1CHRM1PDK1PDK2
SCHEMBL9761867 0.84 HRH1 (0.42) KCNH2HRH1HTR2A
SCHEMBL9762432 0.75 KCNH2 (0.49) KCNH2HRH1CHRM1CYP2D6LSS
SCHEMBL9761690 0.75 KCNH2 (0.49) KCNH2HRH1CHRM1CYP2D6LSS
SCHEMBL9761330 0.75 KCNH2 (0.49) KCNH2HRH1CHRM1CYP2D6LSS
SCHEMBL22130572 0.72 HRH1 (0.36) KCNH2HRH1
SCHEMBL17001812 0.72 HRH1 (0.37) KCNH2HRH1PDK1PDK2PDK3
SCHEMBL25724487 0.69 ALDH1A1 (0.38)
SCHEMBL10446087 0.68 HRH4 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5071855-A Antihistamines, antiallergens DOMPE FARMACEUTICI SPA (IT) 1991-12-10 US disclosed
EP-0397614-A2 Pharmacologically active piperdinylimidazopyridines DOMPE' FARMACEUTICI S.p.A. (IT) 1990-11-14 EP disclosed