SCHEMBL9764393

SCHEMBL9764393

CNC(=O)c1ccc2[nH]cc(C3=CCNCC3)c2c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.59
ALDH1A1 P00352 3/20 0.59
HTR2C P28335 3/20 0.59
HSD17B10 Q99714 3/20 0.59
HTR1D P28221 3/20 0.59
HTR6 P50406 2/20 0.59
MAPT P10636 2/20 0.59
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
CYP1A2 P05177 1/20 0.59
CYP3A4 P08684 1/20 0.59
MAPK1 P28482 1/20 0.59
BRCA1 P38398 1/20 0.59
DRD2 P14416 1/20 0.54
ALOX15 P16050 1/20 0.54
CCNT1 O60563 3/20 0.50
CDK9 P50750 3/20 0.50
JAK2 O60674 1/20 0.49
PRKD3 O94806 1/20 0.49
MARK3 P27448 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558613 0.86 HTR6 (0.65) KDM4EALDH1A1HTR2CHSD17B10HTR1D
SCHEMBL6631360 0.84 HTR6 (0.60) KDM4EALDH1A1HTR2CHSD17B10HTR1D
SCHEMBL8820109 0.82 HSD17B10 (0.56) KDM4EALDH1A1HTR2CHSD17B10HTR1D
SCHEMBL9764510 0.80 SLC6A4 (0.65)
SCHEMBL7487134 0.79 KDM4E (0.65) KDM4EALDH1A1HTR2CHSD17B10HTR1D
SCHEMBL7487825 0.78 HTR6 (0.51) KDM4EALDH1A1HTR2CHSD17B10HTR1D
SCHEMBL24670856 0.78 CCNT1 (0.66) HTR2CHTR6CCNT1CDK9
SCHEMBL29961028 0.78 CCNT1 (0.66) HTR2CHTR6CCNT1CDK9
SCHEMBL3836149 0.77 HTR6 (0.67) KDM4EALDH1A1HTR2CHSD17B10HTR1D
SCHEMBL6631651 0.77 KDM4E (0.70) KDM4EALDH1A1HTR2CHSD17B10HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5066660-A INDOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 1991-11-19 US disclosed
EP-0303506-A2 Indole derivatives GLAXO GROUP LIMITED (GB) 1989-02-15 EP disclosed