SCHEMBL8820109

SCHEMBL8820109

O=C(NCc1ccccc1)c1ccc2[nH]cc(C3=CCNCC3)c2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.56
ALDH1A1 P00352 3/20 0.56
KDM4E B2RXH2 2/20 0.56
MAPT P10636 2/20 0.56
HTR2C P28335 2/20 0.56
DRD2 P14416 1/20 0.56
ALOX15 P16050 1/20 0.56
HTR1D P28221 3/20 0.52
HTR1B P28222 1/20 0.52
HTR6 P50406 2/20 0.50
MAPK1 P28482 2/20 0.49
MEN1 O00255 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
BRCA1 P38398 1/20 0.49
KMT2A Q03164 1/20 0.49
MAPK3 P27361 1/20 0.45
IMPDH2 P12268 1/20 0.44
HPGD P15428 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9764393 0.82 KDM4E (0.59) HSD17B10ALDH1A1KDM4EMAPTHTR2C
Hydrochloric Acid SCHEMBL9764420 0.81 NOS3 (0.59) HSD17B10KDM4EALOX15HTR6
SCHEMBL6631360 0.78 HTR6 (0.60) HSD17B10ALDH1A1KDM4EMAPTHTR2C
SCHEMBL8558613 0.78 HTR6 (0.65) HSD17B10ALDH1A1KDM4EMAPTHTR2C
SCHEMBL5705100 0.74 KDM4E (0.66) HSD17B10ALDH1A1KDM4EMAPTHTR2C
SCHEMBL29379037 0.74 KDM4E (1.00) HSD17B10ALDH1A1KDM4EMAPTHTR2C
SCHEMBL653742 0.74 KDM4E (1.00) HSD17B10ALDH1A1KDM4EMAPTHTR2C
SCHEMBL13533314 0.73 HTR6 (0.63) HSD17B10ALDH1A1KDM4EMAPTHTR2C
SCHEMBL7392593 0.73 JAK2 (0.69) HSD17B10ALDH1A1KDM4EMAPTHTR2C
SCHEMBL7487825 0.73 HTR6 (0.51) HSD17B10ALDH1A1KDM4EMAPTHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997038692-A1 BISINDOLES FOR TREATING PAIN OR NOCICEPTION ELI LILLY AND COMPANY (US) 1997-10-23 WO disclosed