SCHEMBL9765461

SCHEMBL9765461

CCC1(CC)C=Cc2cc(C#N)ccc2O1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
XDH P47989 1/20 0.37
ABCB1 P08183 11/20 0.35
KCNE1 P15382 3/20 0.35
KCNQ1 P51787 3/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35
KCND3 Q9UK17 1/20 0.35
CYP2A6 P11509 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8534981 0.84 CA12 (0.40) CA12CA9PTGS1PTGS2XDH
SCHEMBL30523681 0.80 CA12 (0.46) CA12CA9PTGS1PTGS2XDH
SCHEMBL506743 0.80 CA12 (0.46) CA12CA9PTGS1PTGS2XDH
SCHEMBL9206139 0.74 CA12 (0.40) CA12CA9PTGS1PTGS2XDH
SCHEMBL6980284 0.74 CA12 (0.40) CA12CA9PTGS1PTGS2XDH
SCHEMBL9736524 0.74 PTGS1 (0.46) CA12CA9PTGS1PTGS2XDH
SCHEMBL10511983 0.72 HTR2C (0.45) PTGS1PTGS2XDHMEN1KMT2A
SCHEMBL9876173 0.72 HTR2C (0.49) CA12CA9ABCB1
SCHEMBL7298872 0.72 KCNE1 (0.37) CA12CA9ABCB1KCNE1KCNQ1
SCHEMBL20766474 0.70 ODC1 (0.44) CA12CA9XDHABCB1KCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5071871-A Pharmaceutically useful benzo(β)pyranes and pyranopyridines SANDOZ LTD. (CH) 1991-12-10 US disclosed
US-4988723-A Hypotensive agents, vasodilation FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-01-29 US disclosed
CN-1038811-A 1-benzopyran derivatives and preparation method thereof FUJISAWA PHARMACEUTICAL CO (JP) 1990-01-17 CN disclosed
EP-0344747-A1 Benzopyran derivatives and processes for preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1989-12-06 EP disclosed