SCHEMBL9766043

SCHEMBL9766043

Fc1ccc(CCN2CCN(c3ncc(F)cn3)CC2)cc1

nearest known ligand 0.82

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.82
DRD2 P14416 2/20 0.64
HTR1A P08908 2/20 0.64
DRD1 P21728 1/20 0.64
DRD5 P21918 1/20 0.64
HTR2A P28223 1/20 0.64
DRD3 P35462 1/20 0.64
KDM4E B2RXH2 2/20 0.60
CYP1A2 P05177 1/20 0.60
GAA P10253 1/20 0.60
CYP2C9 P11712 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9765984 0.90 SIGMAR1 (1.00) SIGMAR1DRD2HTR1ADRD1DRD5
Hydrochloric Acid SCHEMBL9766013 0.79 SIGMAR1 (0.60) SIGMAR1DRD2HTR1AHTR2ADRD3
SCHEMBL9766026 0.78 SIGMAR1 (1.00) SIGMAR1DRD2HTR1ADRD1DRD5
SCHEMBL7210648 0.78 SIGMAR1 (0.58) SIGMAR1DRD2HTR1AKDM4ECYP1A2
SCHEMBL9765998 0.76 SIGMAR1 (1.00) SIGMAR1DRD2HTR1ADRD1DRD5
SCHEMBL9602967 0.76 SIGMAR1 (0.79) SIGMAR1DRD2KDM4ECYP1A2GAA
Bmy-14802 SCHEMBL8457738 0.75 SIGMAR1 (1.00) SIGMAR1DRD2DRD3KDM4ECYP1A2
Bmy-14802 SCHEMBL467229 0.75 SIGMAR1 (1.00) SIGMAR1DRD2DRD3KDM4ECYP1A2
SCHEMBL5745400 0.75 KCNJ1 (0.61) SIGMAR1HTR2ACYP1A2
SCHEMBL7855443 0.75 SIGMAR1 (0.63) SIGMAR1DRD2HTR1AKDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4994460-A Treatment or prevention of disorders resulting from central nervous system anoxia BRISTOL-MYERS SQUIBB CO. (US) 1991-02-19 US claimed
EP-0400661-A1 Agents for treatment of brain ischemia Bristol-Myers Squibb Company (US) 1990-12-05 EP claimed