SCHEMBL9767784

SCHEMBL9767784

CN(C(=O)Cc1ccc2ccccc2c1)C1c2ccccc2CC1N1CCCC1

nearest known ligand 0.66

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 11/20 0.66
OPRK1 P41145 7/20 0.63
OPRM1 P35372 6/20 0.63
OPRD1 P41143 3/20 0.63
TP53 P04637 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
TSHR P16473 2/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
MTOR P42345 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 1/20 0.46
MAPK8 P45983 1/20 0.46
MAPK9 P45984 1/20 0.46
MAPK10 P53779 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9767748 0.99 SIGMAR1 (0.65) SIGMAR1OPRK1OPRM1OPRD1TP53
SCHEMBL9643179 0.87 OPRK1 (0.82) SIGMAR1OPRK1OPRM1OPRD1TP53
SCHEMBL7962880 0.87 OPRK1 (0.82) SIGMAR1OPRK1OPRM1OPRD1TP53
SCHEMBL9772344 0.86 SIGMAR1 (0.61) SIGMAR1OPRK1OPRM1OPRD1TP53
Hydrochloric Acid SCHEMBL7077496 0.86 OPRK1 (0.82) SIGMAR1OPRK1OPRM1OPRD1TP53
SCHEMBL7963740 0.86 OPRK1 (0.81) SIGMAR1OPRK1OPRM1OPRD1TP53
Hydrochloric Acid SCHEMBL9813887 0.86 OPRK1 (0.82) SIGMAR1OPRK1OPRM1OPRD1TP53
SCHEMBL9772623 0.86 SIGMAR1 (0.61) SIGMAR1OPRK1OPRM1OPRD1ALDH1A1
SCHEMBL9772473 0.86 OPRK1 (0.81) SIGMAR1OPRK1OPRM1OPRD1TP53
SCHEMBL5632066 0.83 SIGMAR1 (0.57) SIGMAR1OPRK1OPRM1OPRD1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0272982-B1 INDANE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND INTERMEDIATES OBTAINED, THEIR USE AS MEDICINES AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1991-04-17 EP disclosed
US-4988727-A Cardiovascular disorders, analgesics ROUSSEL UCLAF (FR) 1991-01-29 US disclosed
US-4888355-A Indanes and their use as antiarrhythmic agents ROUSSEL UCLAF (FR) 1989-12-19 US disclosed
EP-0272982-A2 Indane derivatives, process for their preparation and intermediates obtained, their use as medicines and compositions containing them ROUSSEL-UCLAF (FR) 1988-06-29 EP disclosed