Bromide

Bromide

SCHEMBL9768264

Br.N=C(N)SCc1cnn(-c2c(Cl)cc(C(F)(F)F)cc2Cl)n1

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.41
ALDH1A1 P00352 5/20 0.38
ALDH2 P05091 4/20 0.38
ALDH3A1 P30838 4/20 0.38
GABRB3 P28472 8/20 0.37
GABRP O00591 7/20 0.37
GABRD O14764 7/20 0.37
GABRA1 P14867 7/20 0.37
GABRB1 P18505 7/20 0.37
GABRG2 P18507 7/20 0.37
GABRA5 P31644 7/20 0.37
GABRA3 P34903 7/20 0.37
GABRA2 P47869 7/20 0.37
GABRB2 P47870 7/20 0.37
GABRA4 P48169 7/20 0.37
GABRE P78334 7/20 0.37
GABRA6 Q16445 7/20 0.37
GABRG1 Q8N1C3 7/20 0.37
GABRG3 Q99928 7/20 0.37
GABRQ Q9UN88 7/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9394102 0.80 GABRB3 (0.44) GABRB3GABRPGABRDGABRA1GABRB1
SCHEMBL9768087 0.79 P2RX7 (0.43) ALDH1A1GABRB3GABRPGABRDGABRA1
SCHEMBL9768155 0.78 GABRA2 (0.39) GABRB3GABRPGABRDGABRA1GABRB1
SCHEMBL9768229 0.78 GABRA2 (0.41) GABRB3GABRPGABRDGABRA1GABRB1
SCHEMBL9768341 0.77 GABRA2 (0.40) GABRB3GABRPGABRDGABRA1GABRB1
SCHEMBL9217807 0.76 GABRA2 (0.41) GABRB3GABRPGABRDGABRA1GABRB1
SCHEMBL9219663 0.76 GABRB3 (0.44) GABRB3GABRPGABRDGABRA1GABRB1
SCHEMBL9219343 0.75 GABRA2 (0.40) ALDH1A1GABRB3GABRPGABRDGABRA1
Methane SCHEMBL27278091 0.75 GABRA2 (0.40) GABRB3GABRPGABRDGABRA1GABRB1
SCHEMBL9501605 0.73 SMN1; SMN2 (0.40) ALDH1A1GABRB3GABRPGABRDGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5064844-A Miticides SCHERING AGROCHEMICALS LIMITED (GB) 1991-11-12 US disclosed
CN-1039345-A TRIAZOLE INSECTICIDES SCHERING AGROCHEMICALS LTD (GB) 1990-02-07 CN disclosed