SCHEMBL9768422

SCHEMBL9768422

O=c1[nH]c2cc(O)ccc2c2oc3ccccc3c12

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 5/20 0.50
CDK5R1 Q15078 4/20 0.50
MAOA P21397 4/20 0.50
DYRK1A Q13627 3/20 0.49
GSK3A P49840 2/20 0.49
GSK3B P49841 2/20 0.49
KDM4E B2RXH2 3/20 0.49
MEN1 O00255 3/20 0.49
HPGD P15428 3/20 0.49
KMT2A Q03164 3/20 0.49
GAA P10253 2/20 0.49
MAPT P10636 2/20 0.49
RECQL P46063 2/20 0.49
BLM P54132 2/20 0.49
ESR2 Q92731 2/20 0.49
MGAM O43451 1/20 0.49
NR1I2 O75469 1/20 0.49
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
ESR1 P03372 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3888726 0.90 CDK5 (0.61) CDK5CDK5R1MAOADYRK1AGSK3A
SCHEMBL9781515 0.89 CDK5 (0.64) CDK5CDK5R1MAOADYRK1AGSK3A
SCHEMBL10664986 0.89 CDK5 (0.52) CDK5CDK5R1MAOADYRK1AGSK3A
SCHEMBL31506760 0.89 CDK5 (0.52) CDK5CDK5R1MAOADYRK1AGSK3A
SCHEMBL9768431 0.84 MAP3K11 (0.49) MAOAKDM4EMEN1HPGDKMT2A
SCHEMBL9781510 0.82 MAOA (0.51) CDK5CDK5R1MAOADYRK1AGSK3A
SCHEMBL9781435 0.81 ESR2 (0.56) CDK5CDK5R1MAOADYRK1AGSK3A
SCHEMBL9781428 0.80 CDK5 (0.62) CDK5CDK5R1MAOADYRK1AGSK3A
SCHEMBL148273 0.80 LMNA (0.49) CDK5CDK5R1MAOADYRK1AGSK3A
SCHEMBL31506767 0.80 MAPT (0.50) KDM4EMEN1HPGDKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2142793-A None JP disclosed
JP-2142792-A None JP disclosed
JP-63297325-A None JP disclosed
US-5073553-A Treatment or prevention of osteoporosis KISSEI PHARMACEUTICAL CO., LTD. (JP) 1991-12-17 US disclosed
US-5023261-A Inhibits bone resorption, stimulates bone hardening and growth KISSEI PHARMACEUTICAL CO., LTD. (JP) 1991-06-11 US disclosed
JP-H02142792-A NOVEL BENZOFUROQUINOLINE DERIVATIVE KISSEI PHARMACEUT CO LTD 1990-05-31 JP disclosed
JP-H02142793-A NOVEL BENZOFUROQUINOLINE DERIVATIVE KISSEI PHARMACEUT CO LTD 1990-05-31 JP disclosed
EP-0370760-A2 Benzofuro[3,2-c]quinoline compounds Kissei Pharmaceutical Co., Ltd. (JP) 1990-05-30 EP disclosed
EP-0357172-A2 Benzofuro[3,2-c]Quinoline compounds Kissei Pharmaceutical Co., Ltd. (JP) 1990-03-07 EP disclosed
JP-S63297325-A REMEDY FOR OSTEOPOROSIS KISSEI PHARMACEUT CO LTD 1988-12-05 JP disclosed
EP-0293146-A1 Benzofuro [3,2-c] quinoline compounds Kissei Pharmaceutical Co. Ltd. (JP) 1988-11-30 EP disclosed