SCHEMBL9768797

SCHEMBL9768797

CCCC(=NN)c1ccncc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
CYP3A4 P08684 2/20 0.38
MPO P05164 1/20 0.38
CYP1A2 P05177 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2A6 P11509 1/20 0.38
CYP2C19 P33261 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
NAAA Q02083 1/20 0.37
KMT2A Q03164 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
GAA P10253 1/20 0.36
NOS3 P29474 2/20 0.36
NOS1 P29475 2/20 0.36
NOS2 P35228 2/20 0.36
CA9 Q16790 1/20 0.35
LMNA P02545 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9768869 0.89 HDAC3 (0.41) KDM4ECYP3A4MPOCYP1A2ADORA3
SCHEMBL9769034 0.84 ATM (0.42) KDM4ECYP3A4MPOCYP1A2ADORA3
SCHEMBL11072536 0.82 GPBAR1 (0.43) KDM4ECYP3A4MPOCYP1A2ADORA3
SCHEMBL9208536 0.80 SMN1; SMN2 (0.53) KDM4EKMT2ASMN1; SMN2NPSR1ALDH1A1
SCHEMBL13317137 0.80 SMN1; SMN2 (0.53) KDM4EKMT2ASMN1; SMN2NPSR1ALDH1A1
SCHEMBL9768970 0.78 KMT2A (0.40) KDM4ECYP3A4MPOCYP1A2ADORA3
SCHEMBL9768946 0.76 GPBAR1 (0.38) KDM4ECYP3A4MPOCYP1A2ADORA3
SCHEMBL9795943 0.73 SMN1; SMN2 (0.57) KDM4ECYP3A4CYP1A2CYP2D6CYP2C19
SCHEMBL9795947 0.73 SMN1; SMN2 (0.57) KDM4ECYP3A4CYP1A2CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL9795925 0.72 SMN1; SMN2 (0.56) KDM4ECYP3A4CYP1A2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5011932-A Anthelmintic pyridinyl acylhydrazones derivatives UPJOHN COMPANY (US) 1991-04-30 US claimed
EP-0214158-A1 ANTHELMINTIC PYRIDINYL ACYLHYDRAZONES, METHOD OF USE AND COMPOSITIONS THE UPJOHN COMPANY (US) 1987-03-18 EP claimed
WO-1986004582-A1 ANTHELMINTIC PYRIDINYL ACYLHYDRAZONES, METHOD OF USE AND COMPOSITIONS THE UPJOHN COMPANY (US) 1986-08-14 WO claimed