SCHEMBL9769034

SCHEMBL9769034

CCC(=NN)c1ccncc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.42
KDM4E B2RXH2 2/20 0.41
MPO P05164 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2A6 P11509 1/20 0.41
CYP2C19 P33261 1/20 0.41
NOS3 P29474 2/20 0.38
NOS1 P29475 2/20 0.38
NOS2 P35228 2/20 0.38
GPBAR1 Q8TDU6 1/20 0.38
KMT2A Q03164 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
NAPRT Q6XQN6 1/20 0.37
LMNA P02545 3/20 0.36
MAPT P10636 3/20 0.36
GAA P10253 3/20 0.36
HPGD P15428 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9768797 0.84 KDM4E (0.38) KDM4EMPOCYP1A2CYP3A4ADORA3
SCHEMBL9768869 0.81 HDAC3 (0.41) KDM4EMPOCYP1A2CYP3A4ADORA3
SCHEMBL2777197 0.81 GPBAR1 (0.49) ATMKDM4EMPOCYP1A2CYP3A4
SCHEMBL2777195 0.81 GPBAR1 (0.49) ATMKDM4EMPOCYP1A2CYP3A4
SCHEMBL9768946 0.79 GPBAR1 (0.38) KDM4EMPOCYP1A2CYP3A4ADORA3
SCHEMBL18193546 0.78 ATM (0.68) ATMKDM4EKMT2ANPSR1LMNA
SCHEMBL9768781 0.77 CYP19A1 (0.47) KDM4ECYP3A4CYP2C19NPSR1MAPT
SCHEMBL13069806 0.76 GSK3B (0.44) ATMKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL28751451 0.73 CTSL (0.50) ATM
SCHEMBL9768868 0.73 GAA (0.49) CYP1A2CYP3A4CYP2D6CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5011932-A Anthelmintic pyridinyl acylhydrazones derivatives UPJOHN COMPANY (US) 1991-04-30 US claimed
EP-0214158-A1 ANTHELMINTIC PYRIDINYL ACYLHYDRAZONES, METHOD OF USE AND COMPOSITIONS THE UPJOHN COMPANY (US) 1987-03-18 EP claimed
WO-1986004582-A1 ANTHELMINTIC PYRIDINYL ACYLHYDRAZONES, METHOD OF USE AND COMPOSITIONS THE UPJOHN COMPANY (US) 1986-08-14 WO claimed
US-5023334-A Anthelmintic pyridinyl acylhydrazones THE UPJOHN COMPANY (US) 1991-06-11 US disclosed
US-5011932-A Anthelmintic pyridinyl acylhydrazones derivatives UPJOHN COMPANY (US) 1991-04-30 US disclosed
EP-0214158-A1 ANTHELMINTIC PYRIDINYL ACYLHYDRAZONES, METHOD OF USE AND COMPOSITIONS THE UPJOHN COMPANY (US) 1987-03-18 EP disclosed
WO-1986004582-A1 ANTHELMINTIC PYRIDINYL ACYLHYDRAZONES, METHOD OF USE AND COMPOSITIONS THE UPJOHN COMPANY (US) 1986-08-14 WO disclosed