SCHEMBL9774749

SCHEMBL9774749

Fc1ccc(OCC2CO2)c(Br)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
PKM P14618 2/20 0.50
GLA P06280 1/20 0.50
TP53 P04637 3/20 0.45
TSHR P16473 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
HIF1A Q16665 2/20 0.45
CYP3A4 P08684 1/20 0.45
TDP1 Q9NUW8 1/20 0.42
RAB9A P51151 2/20 0.40
MAPT P10636 4/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
HTR2A P28223 2/20 0.39
HTR2C P28335 2/20 0.39
HTR2B P41595 2/20 0.39
DRD4 P21917 1/20 0.39
HPGD P15428 2/20 0.37
MEN1 O00255 1/20 0.37
CYP1A2 P05177 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29847319 0.89 ALDH1A1 (0.51) ALDH1A1PKMGLATP53TSHR
SCHEMBL11741482 0.88 ALDH1A1 (0.45) ALDH1A1PKMGLATP53TSHR
SCHEMBL30524198 0.83 ALDH1A1 (0.49) ALDH1A1PKMGLATP53TSHR
SCHEMBL4892470 0.83 ALDH1A1 (0.49) ALDH1A1PKMGLATP53TSHR
SCHEMBL6075086 0.83 ALDH1A1 (0.53) ALDH1A1PKMGLATP53TSHR
SCHEMBL31710828 0.83 PKM (0.49) ALDH1A1PKMSMN1; SMN2RAB9AMAPT
SCHEMBL10407181 0.81 ALDH1A1 (0.49) ALDH1A1PKMGLATP53TSHR
SCHEMBL10407182 0.81 ALDH1A1 (0.46) ALDH1A1PKMGLATP53TSHR
SCHEMBL1044544 0.81 ALDH1A1 (0.50) ALDH1A1PKMGLATP53TSHR
SCHEMBL21296293 0.81 ALDH1A1 (0.50) ALDH1A1GLATP53TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5010198-A Intermediates for the synthesis of benzoxazol- and benzothiazolamine derivatives, useful as anti-anoxic agents JANSSEN PHARMACEUTICA N.V. (BE) 1991-04-23 US disclosed
EP-0184257-B1 BENZOXAZOL- AND BENZOTHIAZOLAMINE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1990-07-25 EP disclosed
US-4861785-A Benzoxazol-and benzothiazolamine derivatives, useful as anti-anoxic agents JANSSEN PHARMACEUTICA N.V. (BE) 1989-08-29 US disclosed
EP-0184257-A1 Benzoxazol- and benzothiazolamine derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1986-06-11 EP disclosed