SCHEMBL9775800

SCHEMBL9775800

Cc1[nH]cnc1CCC(OC(=O)/C=C\C(=O)O)c1cccc(-c2ccccc2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.40
HTR3A P46098 3/20 0.36
HTR3E A5X5Y0 2/20 0.36
HTR3B O95264 2/20 0.36
HTR3D Q70Z44 2/20 0.36
HTR3C Q8WXA8 2/20 0.36
GABRR1 P24046 1/20 0.35
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
RAB9A P51151 1/20 0.34
CTSA P10619 4/20 0.34
F2 P00734 1/20 0.32
CTSL P07711 1/20 0.32
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
PPARG P37231 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL9656231 0.77 HTR3A (0.47) HTR3AHTR3EHTR3BHTR3DHTR3C
Fumaric Acid SCHEMBL9656237 0.77 HTR3A (0.47) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL9775797 0.77 PPARG (0.36) HTR3AHTR3EHTR3BHTR3DHTR3C
Maleic Acid SCHEMBL9657342 0.70 HTR3E (0.53) HTR3AHTR3EHTR3BHTR3DHTR3C
Fumaric Acid SCHEMBL9657347 0.70 HTR3E (0.53) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL9419971 0.68 HCAR2 (0.60) HCAR2ALDH1A1CYP3A4TSHRCYP2C19
SCHEMBL9419967 0.68 HCAR2 (0.60) HCAR2ALDH1A1CYP3A4TSHRCYP2C19
SCHEMBL9420058 0.68 HCAR2 (0.60) HCAR2ALDH1A1CYP3A4TSHRCYP2C19
Maleic Acid SCHEMBL9656108 0.66 HTR3E (0.47) HTR3AHTR3EHTR3BHTR3DHTR3C
Maleic Acid SCHEMBL9656680 0.66 HTR3A (0.54) HTR3AHTR3EHTR3BHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5019586-A 5-Hydroxytryptamine Receptor Antagonists GLAXO GROUP LIMITED 1991-05-28 US disclosed