SCHEMBL9775862

SCHEMBL9775862

CN1CCN(c2cc3nc4c(cc3cc2F)c(=O)c(C(=O)O)cn4C2CC2)CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.55
KDM4E B2RXH2 4/20 0.55
LMNA P02545 3/20 0.55
HPGD P15428 3/20 0.55
HSD17B10 Q99714 2/20 0.55
MAPT P10636 1/20 0.55
CYP1A2 P05177 1/20 0.52
TOP2A P11388 1/20 0.52
CYP2C9 P11712 1/20 0.52
TOP2B Q02880 1/20 0.52
DRD3 P35462 1/20 0.51
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
DPP4 P27487 3/20 0.47
NPC1 O15118 1/20 0.47
PIK3CG P48736 5/20 0.47
PIK3CD O00329 3/20 0.46
PIK3R1 P27986 3/20 0.46
PIK3CA P42336 3/20 0.46
CHRM2 P08172 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9775867 0.90 KDM4E (0.69) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL9775941 0.89 KDM4E (0.56) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL9526209 0.89 KDM4E (0.68) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL9775905 0.88 KDM4E (0.49) ALDH1A1KDM4ELMNAHPGDHSD17B10
Water SCHEMBL9775975 0.88 KDM4E (0.67) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL9775910 0.88 ALDH1A1 (0.46) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL9094359 0.87 ALDH1A1 (0.55) ALDH1A1KDM4ELMNAHPGDHSD17B10
Hydrochloric Acid SCHEMBL9097124 0.86 ALDH1A1 (0.54) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL8941960 0.86 DPP4 (0.49) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL8942340 0.86 DPP4 (0.54) ALDH1A1KDM4ELMNAHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5004745-A Benzo[1,8]naphthyridine derivatives, their preparation and the compositions which contain them LABORATOIRE ROGER BELLON (FR) 1991-04-02 US disclosed
US-4990515-A Chemical intermediates RHONE-POULENC SANTE (FR) 1991-02-05 US disclosed
US-4970213-A Benzo(1,8)naphthyridine derivatives as intermediates RHONE-POULENC SANTE (FR) 1990-11-13 US disclosed