SCHEMBL9775910

SCHEMBL9775910

CCOC(=O)c1cn(C2CC2)c2nc3cc(N4CCN(C)CC4)c(F)cc3cc2c1=O

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.46
KDM4E B2RXH2 7/20 0.46
HPGD P15428 5/20 0.46
HSD17B10 Q99714 4/20 0.46
LMNA P02545 2/20 0.46
MAPT P10636 1/20 0.46
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
ADRB2 P07550 1/20 0.43
DRD3 P35462 1/20 0.42
GAA P10253 1/20 0.41
RAD52 P43351 1/20 0.41
HTT P42858 1/20 0.40
CYP1A2 P05177 1/20 0.40
TOP2A P11388 1/20 0.40
CYP2C9 P11712 1/20 0.40
TOP2B Q02880 1/20 0.40
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8941959 0.89 ADRB2 (0.43) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL9775862 0.88 ALDH1A1 (0.55) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL8942057 0.87 ADRB2 (0.49) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL8941953 0.87 ADRB2 (0.45) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL9775869 0.86 KDM4E (0.47) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7231247 0.84 ADRB2 (0.46) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL9775934 0.84 KMT2A (0.46) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL29576777 0.83 ALDH1A1 (0.66) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL9638922 0.83 ALDH1A1 (0.66) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL8942248 0.83 ADRB2 (0.41) ALDH1A1KDM4EHPGDHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5004745-A Benzo[1,8]naphthyridine derivatives, their preparation and the compositions which contain them LABORATOIRE ROGER BELLON (FR) 1991-04-02 US disclosed
US-4970213-A Benzo(1,8)naphthyridine derivatives as intermediates RHONE-POULENC SANTE (FR) 1990-11-13 US disclosed