SCHEMBL9775902

SCHEMBL9775902

O=C(O)c1cc2cc(F)c(Br)cc2nc1Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.56
NFE2L2 Q16236 1/20 0.56
EGLN1 Q9GZT9 1/20 0.37
STING1 Q86WV6 1/20 0.36
KCNK2 O95069 1/20 0.34
KCNK10 P57789 1/20 0.34
KDM4E B2RXH2 2/20 0.33
DHODH Q02127 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ASPH Q12797 1/20 0.33
KDM8 Q8N371 1/20 0.33
POLB P06746 1/20 0.33
EIF4E P06730 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
HPGD P15428 1/20 0.32
SORT1 Q99523 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30504611 0.87 KEAP1 (0.62) KEAP1NFE2L2STING1KDM4EDHODH
SCHEMBL8889913 0.87 KEAP1 (0.62) KEAP1NFE2L2STING1KDM4EDHODH
SCHEMBL9775865 0.84 KEAP1 (0.59) KEAP1NFE2L2EGLN1STING1KDM4E
SCHEMBL26617507 0.78 KEAP1 (0.54) KEAP1NFE2L2KDM4EDHODHALDH1A1
SCHEMBL21130168 0.76 KDM1A (0.39)
SCHEMBL29911221 0.76 KDM1A (0.39)
SCHEMBL9319284 0.75 KEAP1 (0.50) KEAP1NFE2L2KDM4EALDH1A1MEN1
SCHEMBL2314993 0.74 DHODH (0.48) KEAP1NFE2L2KDM4EDHODHALDH1A1
SCHEMBL22743009 0.74 KEAP1 (0.46) KEAP1NFE2L2KDM4EDHODHALDH1A1
SCHEMBL26632840 0.74 KEAP1 (0.50) KEAP1NFE2L2KDM4EDHODHALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5053509-A Microbiocides; AIDS LABORATOIRE ROGER BELLON (FR) 1991-10-01 US disclosed
US-5004745-A Benzo[1,8]naphthyridine derivatives, their preparation and the compositions which contain them LABORATOIRE ROGER BELLON (FR) 1991-04-02 US disclosed
US-4990515-A Chemical intermediates RHONE-POULENC SANTE (FR) 1991-02-05 US disclosed
US-4970213-A Benzo(1,8)naphthyridine derivatives as intermediates RHONE-POULENC SANTE (FR) 1990-11-13 US disclosed