SCHEMBL9778459

SCHEMBL9778459

CN1CCN(c2nn(S(=O)(=O)c3ccccc3)c3cc(Cl)ccc23)CC1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAT2A P31153 2/20 0.56
HTR6 P50406 11/20 0.53
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
PKM P14618 1/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
POLB P06746 1/20 0.44
DRD2 P14416 3/20 0.43
HTR1A P08908 2/20 0.43
HTR2A P28223 1/20 0.43
ATM Q13315 1/20 0.42
GBA1 P04062 1/20 0.42
DRD1 P21728 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9778470 0.91 HTR6 (0.48) MAT2AHTR6KDM4EALDH1A1GAA
SCHEMBL9778410 0.86 HTR6 (0.48) MAT2AHTR6POLBDRD2HTR1A
SCHEMBL1544859 0.86 HTT (0.43) MAT2AHTR6KDM4EALDH1A1GAA
SCHEMBL1544929 0.86 HTR6 (0.56) HTR6POLBDRD2HTR1AHTR2A
SCHEMBL9778505 0.80 HTR6 (0.48) HTR6HTTPOLBDRD2HTR1A
SCHEMBL9778550 0.78 HTR6 (0.54) HTR6POLBGBA1
SCHEMBL9681923 0.77 MAT2A (0.65) MAT2AHTR6KDM4EALDH1A1GAA
SCHEMBL14140342 0.73 HTR6 (0.54) HTR6POLBDRD2HTR1AHTR2A
SCHEMBL5103496 0.73 HTR6 (0.54) HTR6POLBDRD2HTR1AHTR2A
SCHEMBL5253182 0.73 CNR1 (0.47) HTR6HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4954503-A ANALGESIC, ANTIPSYCHOTIC AGENTS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1990-09-04 US claimed
US-5077405-A Condensation of corresponding phenylsulfonyl compound with condensation agent, cyanation, reduction HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-12-31 US disclosed
EP-0417653-A1 3-(1-Substituted-4-piperazinyl)-1H-indazoles, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-03-20 EP disclosed
US-4954503-A ANALGESIC, ANTIPSYCHOTIC AGENTS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1990-09-04 US disclosed