SCHEMBL9778472

SCHEMBL9778472

CN1CCN(c2nn(C(=O)c3ccccc3)c3ccccc23)CC1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ELANE P08246 8/20 0.51
F2 P00734 2/20 0.51
PLAU P00749 2/20 0.51
RORC P51449 1/20 0.48
HTR3E A5X5Y0 1/20 0.47
HTR3B O95264 1/20 0.47
HTR3A P46098 1/20 0.47
HTR3D Q70Z44 1/20 0.47
HTR3C Q8WXA8 1/20 0.47
SMO Q99835 1/20 0.45
F12 P00748 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9778425 0.86 ELANE (0.46) ELANEHTR3EHTR3BHTR3AHTR3D
SCHEMBL9778381 0.85 SMO (0.44) ELANEHTR3EHTR3BHTR3AHTR3D
SCHEMBL9778473 0.85 MAT2A (0.49) ELANEHTR3ASMO
SCHEMBL10416286 0.83 ELANE (0.56) ELANEF2PLAUSMO
Hydrochloric Acid SCHEMBL9778449 0.82 ELANE (0.55) ELANEF2PLAUSMO
SCHEMBL10395836 0.76 ELANE (0.49) ELANEF2PLAURORC
SCHEMBL10416166 0.76 HTR3E (0.53) HTR3EHTR3BHTR3AHTR3DHTR3C
Hydrochloric Acid SCHEMBL10396434 0.75 ELANE (0.48) ELANEF2PLAURORC
SCHEMBL10415360 0.75 DRD3 (0.49)
Hydrochloric Acid SCHEMBL9778455 0.75 HTR3E (0.51) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4954503-A ANALGESIC, ANTIPSYCHOTIC AGENTS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1990-09-04 US claimed
US-5077405-A Condensation of corresponding phenylsulfonyl compound with condensation agent, cyanation, reduction HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-12-31 US disclosed
EP-0417653-A1 3-(1-Substituted-4-piperazinyl)-1H-indazoles, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-03-20 EP disclosed
US-4954503-A ANALGESIC, ANTIPSYCHOTIC AGENTS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1990-09-04 US disclosed