SCHEMBL9778381

SCHEMBL9778381

CN1CCN(c2nn(C(=O)c3ccccc3)c3cc(F)ccc23)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 2/20 0.44
MAT2A P31153 1/20 0.42
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
HTR3A P46098 1/20 0.41
HTR3D Q70Z44 1/20 0.41
HTR3C Q8WXA8 1/20 0.41
F12 P00748 1/20 0.41
NPC1 O15118 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KMT2A Q03164 1/20 0.40
HTR6 P50406 2/20 0.40
HTT P42858 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
KDM4E B2RXH2 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9778472 0.85 ELANE (0.51) SMOHTR3EHTR3BHTR3AHTR3D
SCHEMBL1545677 0.82 HTR1A (0.43) LMNAHTR6KDM4EALDH1A1
Hydrochloric Acid SCHEMBL1545847 0.81 HTR1A (0.43) LMNAHTR6KDM4EALDH1A1
SCHEMBL10415353 0.81 DRD3 (0.48) LMNARAB9ASMN1; SMN2KMT2AHTR6
SCHEMBL1545439 0.81 KMT2A (0.45) NPC1RAB9AKMT2AMAPK1
Hydrochloric Acid SCHEMBL9778468 0.80 DRD3 (0.47) LMNARAB9ASMN1; SMN2KMT2AHTR6
SCHEMBL9778473 0.79 MAT2A (0.49) SMOMAT2AHTR3ALMNATP53
SCHEMBL9778410 0.78 HTR6 (0.48) MAT2AHTR3EHTR3BHTR3AHTR3D
SCHEMBL9680590 0.78 KHK (0.58) MAT2AHTR3EHTR3BHTR3AHTR3D
Fumaric Acid SCHEMBL8854165 0.78 HTR1A (0.40) LMNAHTR6KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4954503-A ANALGESIC, ANTIPSYCHOTIC AGENTS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1990-09-04 US claimed
US-5077405-A Condensation of corresponding phenylsulfonyl compound with condensation agent, cyanation, reduction HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-12-31 US disclosed
US-4954503-A ANALGESIC, ANTIPSYCHOTIC AGENTS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1990-09-04 US disclosed