SCHEMBL9780183

SCHEMBL9780183

O=S(=O)(c1ccc2c(c1)cc(Br)c1ccccc12)N1CCCNCC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.57
MCOLN3 Q8TDD5 2/20 0.47
TSHR P16473 2/20 0.47
CYP3A4 P08684 3/20 0.46
CYP2D6 P10635 3/20 0.46
MYLK Q15746 3/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
TP53 P04637 2/20 0.46
CYP1A2 P05177 2/20 0.46
NFKB1 P19838 2/20 0.46
MAPK1 P28482 2/20 0.46
CYP2C9 P11712 1/20 0.46
ROCK1 Q13464 3/20 0.46
GMNN O75496 2/20 0.46
LMNA P02545 2/20 0.46
MAPT P10636 2/20 0.46
CYP2C19 P33261 1/20 0.46
MTOR P42345 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6793698 0.80 PKM (0.89) PKMMCOLN3TSHRMEN1KMT2A
Hydrochloric Acid SCHEMBL9780187 0.79 PKM (0.54) PKMMCOLN3TSHRCYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9780283 0.78 PKM (0.79) PKMMCOLN3TSHRMEN1KMT2A
SCHEMBL9094358 0.76 ROCK1 (0.62) PKMMCOLN3TSHRCYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9780189 0.74 PKM (0.54) PKMMCOLN3TSHRCYP3A4CYP2D6
SCHEMBL333988 0.74 PKM (1.00) PKMMCOLN3TSHRMEN1KMT2A
SCHEMBL568043 0.74 ROCK1 (0.60) PKMTSHRCYP3A4CYP2D6MYLK
SCHEMBL6973412 0.74 ALDH1A1 (0.60) PKMTSHRCYP3A4CYP2D6MYLK
Hydrochloric Acid SCHEMBL567792 0.73 ROCK2 (0.61) PKMTSHRCYP3A4CYP2D6MYLK
Hydrochloric Acid SCHEMBL932094 0.73 PKM (0.97) PKMMCOLN3TSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5030631-A Hypotensive, bronchodilator agents SCHERING CORPORATION (US) 1991-07-09 US claimed
US-5030631-A Hypotensive, bronchodilator agents SCHERING CORPORATION (US) 1991-07-09 US disclosed