SCHEMBL9780537

SCHEMBL9780537

CC(Sc1ccc(Cl)cc1Cl)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 3/20 0.50
ITGB2 P05107 2/20 0.44
ICAM1 P05362 2/20 0.44
ITGAL P20701 2/20 0.44
TSHR P16473 3/20 0.44
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
TYMP P19971 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
CASP1 P29466 1/20 0.43
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
AR P10275 1/20 0.41
MRGPRX4 Q96LA9 1/20 0.41
KDM4E B2RXH2 2/20 0.41
LMNA P02545 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9780541 1.00 PPARA (0.50) PPARAITGB2ICAM1ITGALTSHR
SCHEMBL9159642 0.81 ITGB2 (0.45) PPARAITGB2ICAM1ITGALTSHR
SCHEMBL9849304 0.79 RXFP1 (0.49) PPARATYMPSMN1; SMN2ALDH1A1KDM4E
SCHEMBL10652731 0.79 ALDH1A1 (0.55) PPARATSHRALDH1A1
SCHEMBL10651794 0.75 PDE7A (0.51) PPARATSHRSMN1; SMN2ALDH1A1KMT2A
SCHEMBL14644121 0.74 GAA (0.58) TSHRSMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL11295930 0.74 ALDH1A1 (0.40) ITGB2ICAM1ITGALSMN1; SMN2ALDH1A1
SCHEMBL7398296 0.74 CYP2C9 (0.66) PPARATSHRTYMPSMN1; SMN2ALDH1A1
SCHEMBL11518885 0.74 PTGES (0.51) PPARA
SCHEMBL13816918 0.74 ITGB2 (0.46) ITGB2ICAM1ITGALTSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0257378-B1 PYRIMIDINE DERIVATIVES, THEIR PREPARATION AND MEDICAMENTS CONTAINING THESE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1991-07-03 EP disclosed
US-5010060-A Method of treating herpes simplex viral infection employing pyrimidine derivatives HOFFMANN-LA ROCHE INC. (US) 1991-04-23 US disclosed
US-4851519-A AMIDO NUCLEOSIDES, VIRICIDES HOFFMANN-LA ROCHE INC. (US) 1989-07-25 US disclosed
EP-0257378-A1 Pyrimidine derivatives, their preparation and medicaments containing these derivatives F. HOFFMANN-LA ROCHE AG (CH) 1988-03-02 EP disclosed