SCHEMBL9780681

SCHEMBL9780681

Cc1ccc(S(=O)(=O)O)cc1.N#CC(N)C(=O)OCc1ccccc1

nearest known ligand 0.50

Known targets — ChEMBL curated mechanism

ABL1BMXBRAFBTKCHRNA4CHRNB2CSNK1EEGFRERBB2F10FLT1FLT3FLT4IGF1RINSRITKJAK3KDRKITOPRM1PARP1PARP2PDGFRBPIK3CDRAF1RETSLC18A2TECTXKdacAdacBdacCftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.50
MAPT P10636 2/20 0.47
CA1 P00915 6/20 0.43
CA2 P00918 6/20 0.43
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 2/20 0.43
RECQL P46063 2/20 0.43
HPGD P15428 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPK1 P28482 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CTSL P07711 1/20 0.41
CTSK P43235 1/20 0.41
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
PSEN1 P49768 1/20 0.40
PSEN2 P49810 1/20 0.40
APH1B Q8WW43 1/20 0.40
NCSTN Q92542 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670578 0.85 LMNA (0.54) LMNAMAPTCA1CA2ALDH1A1
SCHEMBL716770 0.85 LMNA (0.54) LMNAMAPTCA1CA2ALDH1A1
SCHEMBL719791 0.85 LMNA (0.54) LMNAMAPTCA1CA2ALDH1A1
SCHEMBL5671105 0.85 KMT2A (0.45) LMNACA1CA2ALDH1A1KDM4E
SCHEMBL3528417 0.83 ALDH1A1 (0.50) LMNAALDH1A1CYP2D6MAPK1CYP1A2
SCHEMBL4511022 0.83 LMNA (0.52) LMNAMAPTCA1CA2ALDH1A1
SCHEMBL6890578 0.83 LMNA (0.52) LMNAMAPTCA1CA2ALDH1A1
SCHEMBL6890572 0.83 LMNA (0.52) LMNAMAPTCA1CA2ALDH1A1
SCHEMBL3071 0.83 LMNA (0.52) LMNAMAPTCA1CA2ALDH1A1
SCHEMBL9443648 0.83 LMNA (0.52) LMNAMAPTCA1CA2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5003099-A Method for the production of aminocyanoacetamide LONZA LTD. (CH) 1991-03-26 US disclosed