SCHEMBL8433684

SCHEMBL8433684

CC1CN(c2c(F)cc3c(=O)c(C(=O)O)cn(C4CC4)c3c2Cl)CCN1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.77
KDM4E B2RXH2 7/20 0.77
HPGD P15428 7/20 0.77
KCNH2 Q12809 7/20 0.77
HSD17B10 Q99714 5/20 0.77
POLB P06746 3/20 0.77
OPRM1 P35372 2/20 0.77
PRKD3 O94806 1/20 0.77
ALOX15 P16050 1/20 0.77
CLK2 P49760 1/20 0.77
CLK4 Q9HAZ1 1/20 0.77
TDP1 Q9NUW8 1/20 0.77
CHRM2 P08172 1/20 0.72
CHRM1 P11229 1/20 0.72
OPRD1 P41143 1/20 0.72
PMP22 Q01453 1/20 0.63
HRH3 Q9Y5N1 1/20 0.57
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
LMNA P02545 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10914782 0.99 ALDH1A1 (0.76) ALDH1A1KDM4EHPGDKCNH2HSD17B10
SCHEMBL10654073 0.94 ALDH1A1 (0.70) ALDH1A1KDM4EHPGDKCNH2HSD17B10
SCHEMBL29593740 0.92 ALDH1A1 (0.81) ALDH1A1KDM4EHPGDKCNH2HSD17B10
SCHEMBL6783172 0.92 ALDH1A1 (0.81) ALDH1A1KDM4EHPGDKCNH2HSD17B10
SCHEMBL8435331 0.91 ALDH1A1 (0.66) ALDH1A1KDM4EHPGDKCNH2HSD17B10
SCHEMBL9626969 0.90 ALDH1A1 (0.63) ALDH1A1KDM4EHPGDKCNH2HSD17B10
SCHEMBL3957125 0.90 ALDH1A1 (0.79) ALDH1A1KDM4EHPGDKCNH2HSD17B10
SCHEMBL9792010 0.90 KCNH2 (0.79) ALDH1A1KDM4EHPGDKCNH2HSD17B10
SCHEMBL965845 0.90 ALDH1A1 (0.70) ALDH1A1KDM4EHPGDKCNH2HSD17B10
SCHEMBL10695169 0.90 ALDH1A1 (0.70) ALDH1A1KDM4EHPGDKCNH2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5571812-A TREATMENT OF INFECTIONS OF GRAMNEGATIVE AND GRAMPOSITIVE BACTERIA BAYER AKTIENGESELLSCHAFT (DE) 1996-11-05 US claimed
US-5969141-A Intermediates for 7-amino-1-cyclopropyl-6,8-dihalogeno-1,4-dihydro-4-oxo-3-quinolinecarbox ylic acid antibacterial agents BAYER AKTIENGESELLSCHAFT (DE) 1999-10-19 US disclosed
US-5777181-A 2, 4, 5-trihalogeno- and 2, 3, 4, 5-tetrahalogenobenzene derivatives BAYER AKTIENGESELLSCHAFT (DE) 1998-07-07 US disclosed
US-5571812-A TREATMENT OF INFECTIONS OF GRAMNEGATIVE AND GRAMPOSITIVE BACTERIA BAYER AKTIENGESELLSCHAFT (DE) 1996-11-05 US disclosed
US-5565614-A FLUORINATION BAYER AKTIENGESELLSCHAFT (DE) 1996-10-15 US disclosed
US-5530158-A CHEMICAL INTERMEDIATE FOR ANTIBACTERIALS BAYER AKTIENGESELLSCHAFT (DE) 1996-06-25 US disclosed
US-5468861-A Bactericides BAYER AKTIENGESELLSCHAFT (DE) 1995-11-21 US disclosed
US-5362909-A Two stage fluorination BAYER AKTIENGESELLSCHAFT (DE) 1994-11-08 US disclosed
US-5200548-A Intermediates for bactericides BAYER AKTIENGESELLSCHAFT (DE) 1993-04-06 US disclosed
US-5072038-A Chemical intermediates for bactericides BAYER AKTIENGESELLSCHAFT (DE) 1991-12-10 US disclosed
US-4895803-A QUINOLINE-OR NAPHTHAPYRIDINE/1,8-/ DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 1990-01-23 US disclosed
EP-0191390-B1 1-Cyclopropyl-1,4-dihydro-4-oxo-7-[4-(oxo-1,3-dioxol-4-yl-methyl)-1-piperazinyl]-quinoline-3-carboxylic acids, process for their preparation and bactericides containing them BAYER AG (DE) 1989-08-23 EP disclosed
US-4703047-A 1-Cyclopropyl-1,4-dihydro-4-oxo-7-(4-(2-oxo-1,3-dioxol-4-yl-methyl)-1-piperazinyl)-3-quinolinecarboxylic acid antibacterial agents BAYER AKTIENGESELLSCHAFT (DE) 1987-10-27 US disclosed
EP-0191390-A1 1-Cyclopropyl-1,4-dihydro-4-oxo-7-[4-(oxo-1,3-dioxol-4-yl-methyl)-1-piperazinyl]-quinoline-3-carboxylic acids, process for their preparation and bactericides containing them BAYER AG (DE) 1986-08-20 EP disclosed
EP-0178388-A1 Quinolinecarboxylic acid derivatives KYORIN PHARMACEUTICAL CO., LTD. (JP) 1986-04-23 EP disclosed