SCHEMBL9792939

SCHEMBL9792939

N#Cc1cccc(-c2cc(C#N)ccn2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 3/20 0.62
GRM5 P41594 6/20 0.60
IDO1 P14902 2/20 0.54
CYP1A2 P05177 3/20 0.52
CYP2C19 P33261 3/20 0.52
HSD17B10 Q99714 3/20 0.52
CYP3A4 P08684 2/20 0.52
ALOX15 P16050 1/20 0.52
ASIC3 Q9UHC3 1/20 0.51
MAOB P27338 1/20 0.50
ALDH1A1 P00352 2/20 0.49
USP2 O75604 1/20 0.49
MAPK1 P28482 1/20 0.49
KDM1A O60341 1/20 0.48
XDH P47989 1/20 0.48
GABRA1 P14867 1/20 0.47
GABRG2 P18507 1/20 0.47
GABRB3 P28472 1/20 0.47
GABRA5 P31644 1/20 0.47
GABRA3 P34903 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17116600 0.91 CLK4 (0.51) CLK4GRM5IDO1CYP1A2CYP2C19
SCHEMBL10389736 0.87 CLK4 (0.59) CLK4GRM5IDO1CYP1A2CYP2C19
SCHEMBL30158989 0.87 ASIC3 (0.53) CLK4GRM5CYP1A2CYP2C19HSD17B10
SCHEMBL2949191 0.87 ASIC3 (0.53) CLK4GRM5CYP1A2CYP2C19HSD17B10
SCHEMBL21141650 0.86 CLK4 (0.56) CLK4GRM5IDO1CYP1A2CYP2C19
SCHEMBL17116715 0.86 CLK4 (0.56) CLK4GRM5IDO1CYP1A2CYP2C19
SCHEMBL15344138 0.86 CLK4 (0.56) CLK4GRM5IDO1CYP1A2CYP2C19
SCHEMBL17116421 0.85 CYP11B1 (0.54) CLK4GRM5IDO1CYP1A2CYP2C19
SCHEMBL17116058 0.85 GRM5 (0.47) CLK4GRM5IDO1CYP1A2CYP2C19
SCHEMBL16016610 0.84 GABRG2 (0.63) CLK4GRM5CYP1A2CYP2C19HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5064832-A Bipyrimidine Compounds, Antitumor Agents CIBA-GEIGY CORPORATION (US) 1991-11-12 US disclosed
US-4968804-A Bipyridine compounds CIBA-GEIGY CORPORATION (US) 1990-11-06 US disclosed
EP-0350448-A1 Biaryl compounds CIBA-GEIGY AG (CH) 1990-01-10 EP disclosed