SCHEMBL9794854

SCHEMBL9794854

CCOC(=O)c1ccc(SCCCC(C#N)C(=O)OCC)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.42
CA2 P00918 3/20 0.42
CA12 O43570 2/20 0.42
CA7 P43166 2/20 0.42
CA9 Q16790 2/20 0.42
CA14 Q9ULX7 2/20 0.42
ESR1 P03372 2/20 0.42
ESR2 Q92731 1/20 0.42
LMNA P02545 3/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 1/20 0.41
MAOA P21397 1/20 0.41
HPGD P15428 4/20 0.39
HTT P42858 2/20 0.39
ALDH1A1 P00352 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
HSP90AA1 P07900 1/20 0.39
CACNA1B Q00975 1/20 0.39
APBA1 Q02410 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9794868 0.82 MEN1 (0.52) CA1CA2CA12CA7CA9
SCHEMBL9040146 0.81 CA12 (0.42) CA1CA2CA12CA7CA9
SCHEMBL9794850 0.76 CA1 (0.51) CA1CA2CA12CA7CA9
SCHEMBL9038966 0.76 CA12 (0.51) CA1CA2CA12CA7CA9
SCHEMBL9040642 0.76 CA1 (0.47) CA1CA2CA12CA7CA9
SCHEMBL8982266 0.75 CA1 (0.40) CA1CA2CA12CA7CA9
SCHEMBL9039166 0.74 CYP4A11 (0.52) LMNACYP1A2CYP3A4HPGDHTT
SCHEMBL9343047 0.73 CYP4A11 (0.53) LMNACYP1A2CYP3A4HPGDHTT
SCHEMBL8982245 0.72 TDP1 (0.38) CA1CA2CA12CA7CA9
SCHEMBL9343689 0.72 CYP4A11 (0.52) LMNACYP1A2CYP3A4HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0409382-A1 Glutamic acid derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1991-01-23 EP disclosed
WO-1990014340-A1 GLUTAMIC ACID DERIVATIVES THE WELLCOME FOUNDATION LIMITED (GB) 1990-11-29 WO disclosed
US-4921836-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1990-05-01 US disclosed