SCHEMBL9039166

SCHEMBL9039166

CCOC(=O)C(C#N)CCCc1ccc(C(=O)OC)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4A11 Q02928 3/20 0.52
CYP4F2 P78329 2/20 0.51
LOXL2 Q9Y4K0 1/20 0.42
HTT P42858 1/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
HSD17B10 Q99714 2/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40
ALOX12 P18054 1/20 0.40
CYP2C19 P33261 1/20 0.40
CKS1B P61024 1/20 0.40
SKP2 Q13309 1/20 0.40
HIF1A Q16665 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9343047 0.96 CYP4A11 (0.53) CYP4A11CYP4F2LOXL2HTTKDM4E
SCHEMBL9343689 0.95 CYP4A11 (0.52) CYP4A11CYP4F2LOXL2KDM4EALDH1A1
SCHEMBL11212513 0.84 LOXL2 (0.46) CYP4A11CYP4F2LOXL2HTTKDM4E
SCHEMBL10419232 0.83 PPARA (0.46) KDM4EALDH1A1HPGDTP53CYP1A2
SCHEMBL8982245 0.83 TDP1 (0.38) CYP4A11CYP4F2LOXL2HTTKDM4E
SCHEMBL10480005 0.82 CYP4A11 (0.49) CYP4A11CYP4F2LOXL2HTTKDM4E
SCHEMBL9850083 0.79 DAO (0.34) CYP4A11CYP4F2HTTKDM4EALDH1A1
SCHEMBL10420226 0.79 PPARA (0.44) KDM4EALDH1A1HPGDCYP1A2CYP3A4
SCHEMBL10419972 0.79 PPARA (0.44) KDM4EALDH1A1HPGDCYP1A2CYP3A4
SCHEMBL9050346 0.78 CYP4A11 (0.61) CYP4A11CYP4F2LOXL2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0722440-A1 PYRIMIDINYL-GLUTAMIC ACID DERIVATIVES ELI LILLY AND COMPANY (US) 1996-07-24 EP disclosed
EP-0722440-A4 PYRIMIDINYL-GLUTAMIC ACID DERIVATIVES LILLY CO ELI (US) 1996-06-04 EP disclosed
US-5426110-A Inhibiting dihydrofolate reductase in mammals and treating susceptible reoplasms ELI LILLY AND COMPANY (US) 1995-06-20 US disclosed
WO-1995009845-A1 PYRIMIDINYL-GLUTAMIC ACID DERIVATIVES ELI LILLY AND COMPANY (US) 1995-04-13 WO disclosed
EP-0325343-B1 L-glutamic acid derivatives UNIV PRINCETON (US) 1994-06-22 EP disclosed
US-4871743-A L-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-10-03 US disclosed
EP-0325343-A2 L-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-07-26 EP disclosed