SCHEMBL9796274

SCHEMBL9796274

Cn1cc(OS(C)(=O)=O)c(=O)c2ccc(Cl)cc21

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.41
MAT2A P31153 4/20 0.37
LMNA P02545 1/20 0.36
THRB P10828 1/20 0.36
KDR P35968 1/20 0.36
GSK3B P49841 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 2/20 0.35
MAOB P27338 1/20 0.34
MAPT P10636 1/20 0.34
MAPK8 P45983 1/20 0.34
CYP1A2 P05177 1/20 0.34
ALPL P05186 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9796512 0.89 KMT2A (0.46) GSK3BKMT2AKDM4EMAPTMAPK8
SCHEMBL9796325 0.84 TP53 (0.41) NTRK1LMNATHRBGSK3BKMT2A
SCHEMBL9796539 0.83 CREBBP (0.40) LMNAKMT2AKDM4E
SCHEMBL9796452 0.83 ATM (0.44) GSK3BKMT2AKDM4EMAPK8CYP1A2
SCHEMBL9796276 0.82 ALDH1A1 (0.51) NTRK1GSK3B
SCHEMBL9796185 0.82 KDM4E (0.33) LMNAKMT2AKDM4EMAPTCYP1A2
SCHEMBL9796571 0.80 NR4A2 (0.41) GSK3BMAOB
SCHEMBL9796308 0.80 SCN9A (0.42) MAT2AGSK3BTSHR
SCHEMBL9796435 0.80 PGR (0.45) GSK3BKMT2AMAPTALPL
SCHEMBL6050601 0.80 ALDH1A1 (0.45) LMNAKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997840-A Quinolone sulphonates having antihypertensive activity THE BOOTS COMPANY, PLC (GB) 1991-03-05 US disclosed
EP-0330340-A1 Therapeutic agents The Boots Company PLC (GB) 1989-08-30 EP disclosed
WO-1989007593-A1 THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1989-08-24 WO disclosed