SCHEMBL9796607

SCHEMBL9796607

C=CCc1cccc(-c2ncccn2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.44
CLK4 Q9HAZ1 2/20 0.43
DYRK1A Q13627 1/20 0.43
ADRB2 P07550 1/20 0.43
MAPT P10636 5/20 0.42
LMNA P02545 3/20 0.42
GAA P10253 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MAPK1 P28482 1/20 0.42
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
ALDH1A1 P00352 3/20 0.40
PPARG P37231 2/20 0.40
PPARD Q03181 2/20 0.40
PPARA Q07869 1/20 0.40
XDH P47989 1/20 0.39
KDM4E B2RXH2 2/20 0.38
ALDH2 P05091 1/20 0.38
GABRA1 P14867 1/20 0.38
AKR1B1 P15121 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6850763 0.84 CLK4 (0.44) CLK4DYRK1AADRB2CYP2A6HCRTR1
SCHEMBL13285705 0.83 PTGS2 (0.41) PTGS2MAPTLMNAGAASMN1; SMN2
SCHEMBL29383868 0.82 PTGS2 (0.57) PTGS2MAPTGAASMN1; SMN2MEN1
SCHEMBL5393111 0.82 PTGS2 (0.57) PTGS2MAPTGAASMN1; SMN2MEN1
SCHEMBL29477070 0.82 PTGS2 (0.57) PTGS2MAPTGAASMN1; SMN2MEN1
SCHEMBL9796794 0.81 HRH3 (0.52) PTGS2LMNASMN1; SMN2MAPK1KDM4E
SCHEMBL29725141 0.81 HRH3 (0.52) PTGS2LMNASMN1; SMN2MAPK1KDM4E
SCHEMBL21390635 0.80 KDM4E (0.47) PTGS2MAPTLMNASMN1; SMN2ALDH1A1
SCHEMBL10590683 0.79 ADRB2 (0.57) CLK4ADRB2MAPTLMNAGAA
SCHEMBL6848165 0.79 CLK4 (0.47) CLK4DYRK1AADRB2LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5047172-A W-substituted, optically active alkanol ester derivatives CHISSO CORPORATION (JP) 1991-09-10 US disclosed
EP-0257457-B1 OPTICALLY ACTIVE 2-METHYL 1,3-PROPANEDIOL DERIVATIVES, LIQUID CRYSTAL COMPOSITIONS COMPRISING THEM AND OPTICAL SWITCHING ELEMENT Chisso Corporation (JP) 1990-10-31 EP disclosed
EP-0257457-A2 Optically active 2-methyl 1,3-propanediol derivatives, liquid crystal compositions comprising them and optical switching element Chisso Corporation (JP) 1988-03-02 EP disclosed