SCHEMBL9799749

SCHEMBL9799749

C#Cc1cnc2nc(N)nc(O)c2c1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.35
PIK3CA P42336 4/20 0.34
PIK3CG P48736 4/20 0.34
PIK3CB P42338 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
DHFR P00374 8/20 0.33
MAOA P21397 1/20 0.33
ACHE P22303 1/20 0.33
MAOB P27338 1/20 0.33
EGLN1 Q9GZT9 1/20 0.32
CDK1 P06493 1/20 0.31
CCNB1 P14635 1/20 0.31
MGMT P16455 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
CCNA1 P78396 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9381882 0.75 RARB (0.38) EGLN1
SCHEMBL4072522 0.75 DYRK1B (0.46) PIK3CAPIK3CGDHFR
SCHEMBL13686508 0.75 DHFR (0.43) PIK3CADHFR
SCHEMBL9381296 0.75 IDO1 (0.39) PIK3CAPIK3CGPIK3CBHDAC6DHFR
SCHEMBL9380860 0.73 CYP1A2 (0.37) PARP1EGLN1
SCHEMBL7495317 0.71 ADORA1 (0.39) PARP1EGLN1
SCHEMBL9212955 0.71 DHFR (0.33) PIK3CAPIK3CGDHFR
SCHEMBL9381228 0.68 GABRA1 (0.46) EGLN1
SCHEMBL6305981 0.67 DHFR (0.48) DHFR
SCHEMBL9460321 0.66 DHFR (0.36) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988813-A Process for the preparation of fused pyridine compounds THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-01-29 US disclosed
US-4902796-A 6-alkenyl and ethynyl derivatives of 2-amino-4-hydroxypyrido[2,3-d]pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1990-02-20 US disclosed
US-4818819-A Process for the preparation of fused pyridine compounds THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-04-04 US disclosed
EP-0265126-A2 Process for the preparation of fused pyridine compounds THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1988-04-27 EP disclosed