SCHEMBL9804483

SCHEMBL9804483

N#Cc1ccc(-c2ccc(Oc3ccccc3O)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 3/20 0.53
SLC6A4 P31645 1/20 0.50
AR P10275 1/20 0.50
MMP3 P08254 2/20 0.48
CYP11B2 P19099 1/20 0.45
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
MMP2 P08253 2/20 0.43
POLB P06746 2/20 0.42
PARP15 Q460N3 1/20 0.42
PARP10 Q53GL7 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
GAA P10253 1/20 0.42
IKBKB O14920 1/20 0.42
KDM4E B2RXH2 2/20 0.41
LMNA P02545 2/20 0.41
CYP19A1 P11511 1/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29833728 0.86 CA2 (0.48) ARPOLBGAAIKBKBKDM4E
SCHEMBL8560469 0.86 CA2 (0.48) ARPOLBGAAIKBKBKDM4E
SCHEMBL7700911 0.82 SLC6A4 (0.62) CYP11B1SLC6A4ARCYP11B2PDE4A
SCHEMBL3421695 0.80 SLC6A4 (0.60) CYP11B1SLC6A4ARCYP11B2PDE4A
SCHEMBL29024081 0.80 CA2 (0.54) ARPOLBGAAKDM4ELMNA
SCHEMBL9710755 0.79 CYP11B1 (0.49) CYP11B1SLC6A4ARCYP11B2PDE4A
SCHEMBL24476964 0.78 KDM4E (0.55) SLC6A4MMP3CYP11B2MMP2POLB
SCHEMBL11592335 0.78 CYP19A1 (0.58) SLC6A4MMP3MMP2POLBPARP15
SCHEMBL9344917 0.78 TSHR (0.52) ARPOLBGAAKDM4ELMNA
SCHEMBL7036706 0.77 AR (0.43) CYP11B1SLC6A4ARGAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290591-B1 MATERIALS WITH NITROGENOUS SIX-MEMBERED RINGS MERCK PATENT GmbH (DE) 1991-03-13 EP disclosed
EP-0290591-A1 MATERIALS WITH NITROGENOUS SIX-MEMBERED RINGS. MERCK PATENT GMBH (DE) 1988-11-17 EP disclosed
WO-1988004305-A1 MATERIALS WITH NITROGENOUS SIX-MEMBERED RINGS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1988-06-16 WO disclosed