SCHEMBL9804637

SCHEMBL9804637

CCC(C#N)(Cc1cccnn1)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTDSP1 Q9GZU7 1/20 0.35
CYP1A2 P05177 1/20 0.34
EBP Q15125 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
CCR1 P32246 1/20 0.34
ATM Q13315 1/20 0.33
CYP2D6 P10635 2/20 0.33
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
OPRM1 P35372 1/20 0.33
DRD3 P35462 1/20 0.33
LMNA P02545 1/20 0.33
VNN1 O95497 2/20 0.32
GRIN2B Q13224 4/20 0.31
GRIN1 Q05586 3/20 0.31
CYP3A4 P08684 1/20 0.31
CHRM3 P20309 3/20 0.31
CHRM2 P08172 2/20 0.31
CHRM1 P11229 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9804652 0.80 CTDSP1 (0.32) CTDSP1CYP2D6
SCHEMBL13271382 0.77 CYP2D6 (0.44) EBPSIGMAR1CCR1ATMCYP2D6
SCHEMBL9804889 0.77 CYP1A2 (0.37) CYP1A2EBPSIGMAR1CCR1ATM
SCHEMBL10625675 0.76 ATM (0.47) CYP1A2EBPSIGMAR1CCR1ATM
SCHEMBL9804779 0.75 CCR1 (0.36) CTDSP1EBPSIGMAR1CCR1
SCHEMBL9804758 0.74 CYP2D6 (0.31) CYP2D6
SCHEMBL9804896 0.72 ATM (0.37) CYP1A2EBPSIGMAR1CCR1ATM
SCHEMBL9804906 0.71 CCR1 (0.34) CCR1GRIN2B
SCHEMBL9804854 0.71 CASP1 (0.32) CTDSP1
SCHEMBL11630708 0.68 CCR1 (0.45) EBPSIGMAR1CCR1ATMCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276920-B1 (2-CYANO-2-(PHENYL OR NAPHTHYL)-2-SUBSTITUTED-ETHYL) PYRAZINES, PYRIMIDINES AND PYRIDAZINES ROHM AND HAAS COMPANY (US) 1991-04-03 EP disclosed
EP-0276920-A1 (2-Cyano-2-(phenyl or naphthyl)-2-substituted-ethyl) pyrazines, pyrimidines and pyridazines ROHM AND HAAS COMPANY (US) 1988-08-03 EP disclosed