SCHEMBL9804885

SCHEMBL9804885

CC(C)CCC(C#N)(Cc1cnccn1)c1ccc(F)cc1

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
CYP2D6 P10635 1/20 0.32
HRH1 P35367 1/20 0.32
KCNH2 Q12809 1/20 0.32
TERT O14746 1/20 0.31
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9804704 0.86 KDM4E (0.34) KDM4EALDH1A1HPGDCYP2D6HRH1
SCHEMBL9804803 0.81 CYP19A1 (0.36)
SCHEMBL9804758 0.80 CYP2D6 (0.31) CYP2D6HRH1KCNH2
SCHEMBL9804874 0.77 RORC (0.34) KDM4EALDH1A1HPGDRORC
SCHEMBL9804889 0.72 CYP1A2 (0.37) KDM4ECYP2D6HRH1
SCHEMBL9804872 0.72 TERT (0.38) KDM4EALDH1A1HPGDCYP2D6TERT
SCHEMBL9804810 0.72 CYP19A1 (0.39) KDM4EALDH1A1CYP2D6
SCHEMBL10369963 0.71 CYP19A1 (0.41) CYP2D6KCNH2
SCHEMBL9804742 0.71 CYP19A1 (0.39) KDM4EALDH1A1
SCHEMBL9804805 0.70 CYP19A1 (0.40) KDM4EALDH1A1HPGDTERT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276920-B1 (2-CYANO-2-(PHENYL OR NAPHTHYL)-2-SUBSTITUTED-ETHYL) PYRAZINES, PYRIMIDINES AND PYRIDAZINES ROHM AND HAAS COMPANY (US) 1991-04-03 EP disclosed
EP-0276920-A1 (2-Cyano-2-(phenyl or naphthyl)-2-substituted-ethyl) pyrazines, pyrimidines and pyridazines ROHM AND HAAS COMPANY (US) 1988-08-03 EP disclosed