SCHEMBL980508

SCHEMBL980508

O=C(Nc1cccc(-c2cnn(Cc3ccccc3)c2)c1)c1cc2cccc(O)c2oc1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKE Q14164 2/20 0.48
TBK1 Q9UHD2 2/20 0.48
AKR1C3 P42330 4/20 0.47
CASP3 P42574 1/20 0.47
CBR1 P16152 2/20 0.46
SCD O00767 2/20 0.46
AR P10275 1/20 0.46
SCD5 Q86SK9 1/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
KMT2A Q03164 1/20 0.45
PTK2B Q14289 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
BACE1 P56817 1/20 0.45
AKR1B10 O60218 1/20 0.44
AKR1B1 P15121 1/20 0.44
F12 P00748 3/20 0.44
MAOB P27338 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL980522 0.89 CASP3 (0.61) CASP3NPC1RAB9APOLBMAPT
SCHEMBL981025 0.83 CASP3 (0.51) AKR1C3CASP3CBR1ARNPC1
SCHEMBL978163 0.78 MAOB (0.52) AKR1C3CASP3CBR1ARNPC1
SCHEMBL980408 0.77 KMT2A (0.52) AKR1C3CASP3CBR1ARNPC1
SCHEMBL980671 0.77 MAPK1 (0.55) AKR1C3CASP3CBR1ARNPC1
SCHEMBL979386 0.77 AKR1C3 (0.51) AKR1C3CASP3CBR1ARNPC1
SCHEMBL980848 0.76 CASP3 (0.50) AKR1C3CASP3CBR1ARNPC1
SCHEMBL977891 0.76 AKR1C3 (0.54) AKR1C3CASP3CBR1ARNPC1
SCHEMBL982797 0.75 AKR1C3 (0.59) AKR1C3CBR1ARNPC1RAB9A
SCHEMBL979803 0.75 MAOB (0.51) AKR1C3CASP3CBR1ARNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110021522-A1 ACTIVATORS OF EXECUTIONER PROCASPASES 3, 6 AND 7 THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2011-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110021522-A1 ACTIVATORS OF EXECUTIONER PROCASPASES 3, 6 AND 7 CASP7, CASP3, CASP6 IKBKE 915/4885TBK1 1723/4885AKR1C3 3154/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.