SCHEMBL9808448

SCHEMBL9808448

Cc1csc(C(=O)CCc2ccccc2)c1OCCN(C)C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.43
S1PR3 Q99500 1/20 0.43
ALDH1A1 P00352 4/20 0.42
ABCB1 P08183 3/20 0.41
HRH1 P35367 1/20 0.40
KDM4E B2RXH2 3/20 0.40
EGFR P00533 2/20 0.40
LTA4H P09960 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ATM Q13315 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
DRD2 P14416 1/20 0.39
DRD1 P21728 1/20 0.39
DRD4 P21917 1/20 0.39
DRD5 P21918 1/20 0.39
UTS2R Q9UKP6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10565203 0.99 S1PR1 (0.42) S1PR1S1PR3ALDH1A1ABCB1HRH1
SCHEMBL9808381 0.88 SCN1A (0.44) ALDH1A1ABCB1KDM4EEGFRLTA4H
Hydrochloric Acid SCHEMBL9808512 0.87 SCN1A (0.43) ALDH1A1ABCB1KDM4ELTA4HMEN1
SCHEMBL9808422 0.80 ABCB1 (0.58) ALDH1A1ABCB1KDM4ELTA4H
SCHEMBL9808398 0.79 ABCB1 (0.60) ALDH1A1ABCB1KDM4ELTA4H
Hydrochloric Acid SCHEMBL9808527 0.79 ABCB1 (0.57) ALDH1A1ABCB1LTA4H
Hydrochloric Acid SCHEMBL9808486 0.78 ABCB1 (0.59) ALDH1A1ABCB1KDM4EEGFRLTA4H
SCHEMBL9316458 0.78 MGLL (0.42) ALDH1A1ABCB1NPC1RAB9A
SCHEMBL9808491 0.77 MEN1 (0.56) ALDH1A1ABCB1KDM4EEGFRLTA4H
Hydrochloric Acid SCHEMBL9808395 0.76 ALDH1A1 (0.57) ALDH1A1ABCB1EGFRLTA4HMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0266336-B1 1-[3-(2-Dialkylaminoethoxy)-2-thienyl]-3-phenyl-1-propanones and their acid addition salts, process for their preparation and pharmaceutical compositions containing them Binder, Dieter, Prof. Dr. (AT) 1991-05-15 EP claimed
EP-0266336-A1 1-[3-(2-Dialkylaminoethoxy)-2-thienyl]-3-phenyl-1-propanones and their acid addition salts, process for their preparation and pharmaceutical compositions containing them Binder, Dieter, Prof. Dr. (AT) 1988-05-04 EP claimed
EP-0266336-B1 1-[3-(2-Dialkylaminoethoxy)-2-thienyl]-3-phenyl-1-propanones and their acid addition salts, process for their preparation and pharmaceutical compositions containing them Binder, Dieter, Prof. Dr. (AT) 1991-05-15 EP disclosed
US-4814330-A CARDIOVASCULAR DISORDERS BINDER DIETER (AT) 1989-03-21 US disclosed