SCHEMBL9810146

SCHEMBL9810146

C#CC(C)(O)Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.50
TAAR1 Q96RJ0 1/20 0.50
CYP2C9 P11712 2/20 0.48
CYP2C19 P33261 2/20 0.48
CYP1A2 P05177 2/20 0.48
LMNA P02545 2/20 0.47
CYP2D6 P10635 1/20 0.47
TRPA1 O75762 1/20 0.46
FDPS P14324 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.41
HIF1A Q16665 1/20 0.41
CYP3A4 P08684 3/20 0.40
ALDH1A1 P00352 1/20 0.40
EGFR P00533 1/20 0.39
USP2 O75604 1/20 0.38
TSHR P16473 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
PYCR1 P32322 1/20 0.38
KCNA5 P22460 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17974969 0.85 TAAR1 (0.48) SLC6A2TAAR1CYP2C9CYP2C19CYP1A2
SCHEMBL11224610 0.82 TDP1 (0.40) SLC6A2TAAR1LMNAFDPSALDH1A1
SCHEMBL11043392 0.81 SLC6A2 (0.48) SLC6A2TAAR1CYP2C9CYP2C19CYP1A2
SCHEMBL4528233 0.80 SLC6A2 (0.52) SLC6A2TAAR1CYP2C9CYP2C19CYP1A2
SCHEMBL28756083 0.80 CYP1A2 (0.50) SLC6A2TAAR1CYP2C9CYP2C19CYP1A2
SCHEMBL700506 0.79 PYCR1 (0.42) TAAR1CYP2C9CYP2C19LMNACYP2D6
SCHEMBL4621803 0.79 FDPS (0.47) CYP2C9CYP2C19CYP1A2LMNACYP2D6
SCHEMBL9806913 0.79 SLC6A2 (0.47) SLC6A2TAAR1CYP2C9CYP2C19CYP1A2
SCHEMBL8341995 0.79 CYP19A1 (0.47) SLC6A2TAAR1CYP3A4ALDH1A1MAOA
SCHEMBL10925250 0.79 DRD2 (0.47) TAAR1CYP1A2LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107759478-B Thermosetting polyimide material containing dicarboborane, preparation method and application 北京航空航天大学 2020-07-14 CN disclosed
CN-107759478-A A kind of Thermocurable polyimide material and preparation method and application containing double carboranes 北京航空航天大学 2018-03-06 CN disclosed
EP-0255098-B1 Novel 8-(lower alkyl) bicyclo [4.2.0] octane derivatives with valuable therapeutic properties SYNTEX (U.S.A.) INC. (US) 1991-05-29 EP disclosed
EP-0196617-B1 [4.2.0]bicyclooctane derivatives, process for their preparation and pharmaceutical compositions containing same SYNTEX (U.S.A.) INC. (US) 1989-05-31 EP disclosed
US-4735966-A ANTICOAGULANTS, VASODILATORS, HYPOTENSIVE AND ANTICHOLESTEROL AGENTS SYNTEX (U.S.A.) INC. (US) 1988-04-05 US disclosed
EP-0257609-A2 Novel substituted (4.2.0)Bicyclooctane derivatives with valuable therapeutic properties SYNTEX (U.S.A.) INC. (US) 1988-03-02 EP disclosed
EP-0255098-A1 Novel 8-(lower alkyl) bicyclo [4.2.0] octane derivatives with valuable therapeutic properties SYNTEX (U.S.A.) INC. (US) 1988-02-03 EP disclosed
US-4678805-A Novel 8-(lower alkyl)bicyclo[4.2.0]octane derivatives with valuable therapeutic properties SYNTEX (U.S.A.) INC. (US) 1987-07-07 US disclosed
EP-0196617-A1 [4.2.0]bicyclooctane derivatives, process for their preparation and pharmaceutical compositions containing same SYNTEX (U.S.A.) INC. (US) 1986-10-08 EP disclosed
US-4608388-A Novel [4,2,0]bicyclooctane derivatives with valuable therapeutic properties SYNTEX (U.S.A.) INC. (US) 1986-08-26 US disclosed