SCHEMBL9813079

SCHEMBL9813079

COC(=O)C1CC(c2ccncc2)CCC1=O

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
ROCK2 O75116 7/20 0.37
PRKG1 Q13976 6/20 0.37
LMNA P02545 1/20 0.36
MMP2 P08253 1/20 0.36
ANPEP P15144 1/20 0.36
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9878558 0.87 KDM4E (0.42) PDE3BPDE3ALMNA
SCHEMBL7272419 0.85 PDE3B (0.44) PDE3BPDE3AROCK2PRKG1LMNA
SCHEMBL9543367 0.83 HTT (0.46)
SCHEMBL10665721 0.82 PDE3B (0.39) PDE3BPDE3AROCK2PRKG1LMNA
SCHEMBL10666182 0.81 PDE3B (0.38) PDE3BPDE3AROCK2PRKG1LMNA
SCHEMBL14449885 0.79 SLC6A3 (0.36)
SCHEMBL13920733 0.79 SLC6A3 (0.36)
SCHEMBL13920693 0.79 KDM4E (0.43) LMNADDB1CRBN
SCHEMBL13920699 0.79 HCAR2 (0.39) LMNA
SCHEMBL791422 0.78 MAPK1 (0.41) MMP2ANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5047545-A 2-alkoxycarbonyl-4-(4-pyridyl)cyclohexanones and process for preparing them MITSUI TOATSU CHEMICALS, INC. (JP) 1991-09-10 US claimed
EP-0281661-B1 2-ALKOXYCARBONYL-4-(4-PYRIDYL)CYCLOHEXANONES AND PROCESS FOR PREPARING THEM MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-07-17 EP claimed
CN-87101872-A 2-carbalkoxy-4-(4-pyridyl) pimelinketone and preparation method thereof 1988-09-21 CN claimed
EP-0281661-A1 2-Alkoxycarbonyl-4-(4-pyridyl)cyclohexanones and process for preparing them MITSUI TOATSU CHEMICALS, Inc. (JP) 1988-09-14 EP claimed
US-5047545-A 2-alkoxycarbonyl-4-(4-pyridyl)cyclohexanones and process for preparing them MITSUI TOATSU CHEMICALS, INC. (JP) 1991-09-10 US disclosed
US-5047545-A 2-alkoxycarbonyl-4-(4-pyridyl)cyclohexanones and process for preparing them MITSUI TOATSU CHEMICALS, INC. (JP) 1991-09-10 US disclosed
EP-0281661-B1 2-ALKOXYCARBONYL-4-(4-PYRIDYL)CYCLOHEXANONES AND PROCESS FOR PREPARING THEM MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-07-17 EP disclosed
EP-0281661-A1 2-Alkoxycarbonyl-4-(4-pyridyl)cyclohexanones and process for preparing them MITSUI TOATSU CHEMICALS, Inc. (JP) 1988-09-14 EP disclosed
EP-0281661-A1 2-Alkoxycarbonyl-4-(4-pyridyl)cyclohexanones and process for preparing them MITSUI TOATSU CHEMICALS, Inc. (JP) 1988-09-14 EP disclosed